Target Details
UniProt ACP53667
Gene SymbolLIMK1
Protein NameLIM domain kinase 1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00412 (LIM) PF00595 (PDZ) PF07714 (PK_Tyr_Ser-Thr)
Summary
  • Multi-target molecules 364
  • Clinical molecules 14
  • Avg pChEMBL 7.01
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (364)
InChIKey pChEMBL Type Targets Clinical
FFDIPAAUHNHALW 7.2 IC50 2
UMQNZSBIZJEBSD 7.2 IC50 6
RYXLLTGGHCFCFK 7.2 IC50 3
WTEYHNUOCXPIPD 7.2 Ki 2
PFTXFNSHFZLJNT 7.2 IC50 17
SNLKOFNBEZIHOP 7.2 Ki 2
GXDVQXKUXBTEPR 7.1 Ki 2
ANYTXBDCXZHXLS 7.1 Ki 2
KNACLJBHKVSTDL 7.1 Ki 40
YDOPLCNFRXOHCC 7.1 Ki 28
BAPWDXJBRBPFJX 7.1 Ki 2
CBNCDUSBRPUANI 7.1 Ki 2
XOSKGVORWORZSZ 7.1 Ki 2
NSNKKSURBOMEKE 7.1 IC50 3
XKNKSXHITXPWPU 7.1 IC50 2
IDNMXWIZDRKKBP 7.0 Ki 2
XMUKDUMZYDMRTB 7.0 Ki 2
OOMBFNDWQIGHEK 7.0 Kd 22
UITUOFHXOHTXBO 7.0 Ki 2
WXPPFJWCYWVAFA 7.0 Ki 2
GSHQEEILURASRZ 7.0 Ki 2
NXEVMWHFSSQBGY 7.0 IC50 2
OYYKGCKVVURSQO 7.0 IC50 2
CWTWMAPTTBKMQQ 7.0 IC50 2
HKSZLNNOFSGOKW 7.0 Ki 118
IOBVCHJTLVPPBR 7.0 Ki 39
IXBDAXIRGAZGHU 7.0 Ki 2
JHYHWHUTTXJICB 7.0 Ki 18
KTEIFNKAUNYNJU 7.0 Ki 48
RGNHKJWHFIPHIM 7.0 Ki 66
XKFTZKGMDDZMJI 7.0 Ki 56
NYOZZACQGGCRNW 7.0 Ki 2
RXNNVMXDYOSEDL 7.0 Ki 2
MINOKEADQMWBJE 7.0 Ki 2
QLSVQOIIIVLATL 7.0 Ki 2
CFYUOSYOZDRMJV 6.9 Ki 2
WNJHZIAEDRPGFZ 6.9 Ki 2
XCZSICUSGXTGKT 6.9 IC50 2
ZBNZXTGUTAYRHI 6.9 IC50 102 Yes
OYNRZTXCSUROSS 6.9 IC50 2
IWAGHIAOERSNDT 6.9 IC50 2
NCQISIHBBJLDQW 6.9 Ki 2
GUHUQPHEGAYGKK 6.9 Ki 4
MCCCQFAOMZMZKE 6.9 Ki 52
RYYNGWLOYLRZLK 6.9 Ki 104
YGKFZWJWKPZPQM 6.9 Ki 13
ZCCJKVBTHCOISJ 6.9 Ki 46
SLEWGGZPOQNVSU 6.9 Kd 22
ZDQTUWBKEDTMHG 6.9 Ki 2
YFNWWNRZJGMDBR 6.9 Kd 35
2D structure