Target Details
UniProt ACP53667
Gene SymbolLIMK1
Protein NameLIM domain kinase 1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00412 (LIM) PF00595 (PDZ) PF07714 (PK_Tyr_Ser-Thr)
Summary
  • Multi-target molecules 364
  • Clinical molecules 14
  • Avg pChEMBL 7.01
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (364)
InChIKey pChEMBL Type Targets Clinical
SEZBMVMOFIKXMB 9.5 IC50 2
KSECQYDNQYAZMQ 9.3 IC50 3
YTTBQAOPTOOIMN 9.0 IC50 2
GDVRVPIXWXOKQO 8.8 IC50 10
SCAJVURXKFKCRM 8.6 Ki 2
HCTRFFWHDWFRRD 8.5 Ki 2
MVPARBNSRQJBEM 8.5 IC50 3
RZCBPADGHYZXSD 8.4 IC50 3
BJLGGRFJWDFWQM 8.4 Ki 2
WTRQXHALVSEXHZ 8.4 IC50 3
YROFKBMFSNSLOY 8.3 Ki 2
DWMTZHKJEKZMNU 8.3 Ki 2
XWDRWEDLKSVHEF 8.3 Ki 2
JDJMYZHNJPZTEO 8.3 Ki 2
MPASMALZLVDLOE 8.3 Ki 2
BQBOOEFYJFITIW 8.3 Ki 2
IAMISDYFBNNTFD 8.2 Ki 2
NXSJMRCTGYTSTK 8.2 Kd 200
GZLAHVJYSXFVMI 8.2 Ki 2
KFCPGWYTVYMYJT 8.2 Ki 2
JQXGSDPBFXEDBN 8.2 IC50 4
FWSCHTFTQUFXQK 8.2 Ki 2
ANERHQSYBWTJAR 8.2 Ki 2
CRQMPLKPSNDETC 8.2 Ki 2
JBWCXUIDKXVDBB 8.2 Ki 2
HFBCKXXEXNDPEJ 8.1 IC50 5
QJSHRSRHXNILPU 8.1 Ki 2
UIQNMIISGRIHIY 8.1 IC50 2
PRTHCCVOFVEANA 8.1 Ki 2
JYKZUHVJQBUTEZ 8.1 Ki 2
POHPJJMFSJEVCL 8.0 Ki 2
CGZODTDSSKPGEE 8.0 Ki 2
GKKPPDHQVAOQNK 8.0 Ki 2
HVHFPGDOEVTOET 7.9 Ki 2
FDJOHHPXPWKDPJ 7.9 Ki 2
LBTIFWLBYCBNOX 7.9 Ki 2
PTHVKCSYXICMAR 7.9 IC50 14
BTVPMDAMCUGYJV 7.9 IC50 4
OBRSOISWMBOHDY 7.9 Ki 2
NIASVIHRSPCQKW 7.9 Ki 2
RYYHCXZWRDDPPO 7.9 Ki 2
FYQRHEPZQPVRBM 7.9 Ki 2
MVKANPXDEKJERH 7.8 Ki 2
NHONHQMEURDYOT 7.8 Ki 2
ZHVBPFYLCBVTAE 7.8 Ki 2
ZOJJLNGGZSQITE 7.8 Ki 2
PWUPADCGCCPNFN 7.8 Ki 2
YVPYJSSYGACUSE 7.8 IC50 2
FHOUAZWJJGMZPN 7.8 Ki 2
VWMGMUUIICOGGW 7.8 Ki 2
2D structure