Target Details
| UniProt AC | P53634 |
|---|---|
| Gene Symbol | CTSC |
| Protein Name | Dipeptidyl peptidase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08773 (CathepsinC_exc) PF00112 (Peptidase_C1) |
Summary
- Multi-target molecules 33
- Clinical molecules 1
- Avg pChEMBL 7.5
KEGG Pathways (2)
Associated Diseases (4)
Active Molecules (33)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DTAUFOVRLHTZMV
|
9.1 | IC50 | 2 | — | |
JTEJDGCXJPQUEE
|
9.1 | IC50 | 2 | — | |
MXFQVQKDFVESOP
|
9.0 | IC50 | 2 | — | |
NMLYRXXREIIYKN
|
8.7 | IC50 | 2 | — | |
XOGLUHPWGGYHRM
|
8.7 | IC50 | 4 | — | |
AQJIKVTXFPNTKB
|
8.4 | IC50 | 2 | — | |
NLFOFOVCNGNZSN
|
8.2 | IC50 | 2 | — | |
RYOBYDLUILCXPC
|
8.2 | IC50 | 2 | — | |
XCTNQGKKNUPDFM
|
8.1 | IC50 | 4 | — | |
SRQKADSCZJGWOI
|
8.0 | IC50 | 2 | — | |
ZCCPLJOKGAACRT
|
8.0 | Kd | 599 | — | |
FUYOZZGSCQXNCB
|
7.8 | IC50 | 3 | — | |
FUYOZZGSCQXNCB
|
7.8 | IC50 | 3 | — | |
OWXGOHWYUAIZNU
|
7.8 | IC50 | 2 | — | |
YLYRPDLKZYLBQM
|
7.8 | IC50 | 2 | — | |
SIIJWJNEODXHNY
|
7.7 | IC50 | 7 | — | |
NWEHEPXTNMPJSH
|
7.7 | IC50 | 2 | — | |
ZFTSPYMTXLAPOD
|
7.7 | IC50 | 2 | — | |
GCWIICJLIHIUNY
|
7.5 | IC50 | 7 | — | |
SZYYBVWPURUFRR
|
7.5 | IC50 | 8 | — | |
GLJZTHKUTGOBFU
|
7.1 | IC50 | 4 | — | |
OMZCMEYTWSXEPZ
|
6.9 | IC50 | 43 | Yes | |
OBODFDBEYMKZMM
|
6.9 | IC50 | 2 | — | |
ORFRHRXPOJVPSF
|
6.8 | IC50 | 2 | — | |
YOGVFFRGTMXMRZ
|
6.7 | IC50 | 5 | — | |
FXILBKWGQQHVJE
|
6.5 | IC50 | 3 | — | |
FXILBKWGQQHVJE
|
6.5 | IC50 | 2 | — | |
CFOTUZHUTFRFQA
|
6.4 | IC50 | 5 | — | |
VHNVOAVIDBRLFO
|
6.3 | IC50 | 4 | — | |
VLZYXSQGILGQAI
|
6.2 | IC50 | 6 | — | |
BMIOGAIQRVIVKQ
|
6.2 | IC50 | 4 | — | |
LTLYEAJONXGNFG
|
6.1 | IC50 | 9 | — | |
VHDAHAMWVNXMSP
|
6.1 | IC50 | 7 | — |