Target Details
| UniProt AC | P53609 |
|---|---|
| Gene Symbol | PGGT1B |
| Protein Name | Geranylgeranyl transferase type-1 subunit beta |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00432 (Prenyltrans) |
Summary
- Multi-target molecules 232
- Clinical molecules 172
- Avg pChEMBL 7.05
Active Molecules (232)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UXBVMEPFELTEOC
|
6.2 | IC50 | 3 | — | |
LEOFHPLVHZUFJS
|
6.2 | IC50 | 3 | Yes | |
USPFJPDEADLGIG
|
6.2 | IC50 | 3 | Yes | |
CYBHYVCTXZJLET
|
6.2 | IC50 | 3 | Yes | |
HMBVZGUDIZJMIK
|
6.2 | IC50 | 3 | Yes | |
OAFSUCMIFLKJKF
|
6.2 | IC50 | 3 | — | |
QUQDOQTVANCRAB
|
6.2 | IC50 | 3 | Yes | |
UNMKLZBYJNBEEK
|
6.2 | IC50 | 3 | Yes | |
HRCUJSFALQORGR
|
6.1 | IC50 | 3 | Yes | |
RYKIAQZQXCZXEZ
|
6.1 | IC50 | 3 | Yes | |
PPQXZTKHXAKMSY
|
6.1 | IC50 | 2 | — | |
YHWHZGNJXZQUQM
|
6.1 | IC50 | 5 | — | |
FBTSVHIGWRLBOS
|
6.1 | IC50 | 3 | Yes | |
BDXLTTUQHGMFEE
|
6.1 | IC50 | 3 | Yes | |
HAVQUHAYFMIFJN
|
6.1 | IC50 | 3 | — | |
HYDRIOWWHJJSSW
|
6.1 | IC50 | 3 | Yes | |
MVPXMHNFAQUXRM
|
6.1 | IC50 | 3 | Yes | |
SUHLJVHSQCIBRD
|
6.1 | IC50 | 3 | Yes | |
SQSRCLAOTRHUQX
|
6.1 | IC50 | 3 | Yes | |
GOQKNURHCDAYKJ
|
6.1 | IC50 | 3 | Yes | |
MARYRVHUZOQJMX
|
6.1 | IC50 | 2 | — | |
DIDRALNGAJEZDV
|
6.1 | IC50 | 4 | Yes | |
MRIIEPZJIMUDLC
|
6.1 | IC50 | 3 | Yes | |
SRVLVBDYUWMIOB
|
6.1 | IC50 | 3 | Yes | |
AFXXVFSLJYLSOC
|
6.0 | IC50 | 3 | Yes | |
BHKKLGROGAROGK
|
6.0 | IC50 | 3 | Yes | |
MDOOQICNCKEHFW
|
6.0 | IC50 | 3 | Yes | |
PRLPUFDEFXKPJO
|
6.0 | IC50 | 3 | — | |
IGCOPNHCHHWZNH
|
6.0 | IC50 | 3 | Yes | |
NCOZXTAQUOCINN
|
6.0 | IC50 | 3 | Yes | |
QAJIHSCJMHBCFI
|
6.0 | IC50 | 3 | Yes | |
UMMFUJAKLTXUKT
|
6.0 | IC50 | 3 | Yes |