Target Details
| UniProt AC | P53609 |
|---|---|
| Gene Symbol | PGGT1B |
| Protein Name | Geranylgeranyl transferase type-1 subunit beta |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00432 (Prenyltrans) |
Summary
- Multi-target molecules 232
- Clinical molecules 172
- Avg pChEMBL 7.05
Active Molecules (232)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CKUAWXYQQWMTHM
|
6.5 | IC50 | 3 | Yes | |
LQJGIUPYFFXRBB
|
6.5 | IC50 | 3 | Yes | |
OJEWQHUSLNOLBT
|
6.5 | IC50 | 3 | Yes | |
NLKNPWNNYCYNKB
|
6.5 | IC50 | 3 | Yes | |
HPTPUWFOBXCUAN
|
6.5 | IC50 | 3 | Yes | |
OHMYEZKFMQAYKQ
|
6.5 | IC50 | 5 | — | |
AHPUIZQTTZGXBJ
|
6.5 | IC50 | 3 | Yes | |
UMMFUJAKLTXUKT
|
6.5 | IC50 | 3 | Yes | |
OINNEUNVOZHBOX
|
6.5 | IC50 | 2 | — | |
BYAJXJYFHAJINJ
|
6.5 | IC50 | 3 | Yes | |
SCTKIRVLFRCMEU
|
6.5 | IC50 | 2 | — | |
RLZPEQLIWYHFHH
|
6.4 | IC50 | 3 | Yes | |
SUXXIEYIKBWNGK
|
6.4 | IC50 | 3 | Yes | |
VWNBOOIWICWEPL
|
6.4 | IC50 | 3 | — | |
FTCZIJXHWDHTQT
|
6.4 | IC50 | 2 | — | |
VBOYISMKUMBEJC
|
6.4 | IC50 | 3 | Yes | |
SFKOTJCSIYBZQW
|
6.4 | IC50 | 3 | Yes | |
AQRLDBGCWSEIIY
|
6.4 | IC50 | 3 | Yes | |
CKVSFSCNFUEJNJ
|
6.3 | IC50 | 3 | Yes | |
GSHROJORMPAUBU
|
6.3 | IC50 | 2 | — | |
XKBOADWPZLOLCO
|
6.3 | IC50 | 3 | Yes | |
MWHMRNQLNHVBSC
|
6.3 | IC50 | 2 | — | |
YCUWEXRMZLDWND
|
6.3 | IC50 | 3 | Yes | |
XXNOXIHVPUERGU
|
6.3 | IC50 | 3 | Yes | |
MXROXRMSFVHUHH
|
6.3 | IC50 | 3 | Yes | |
BJSYVDIHBYVMSH
|
6.3 | IC50 | 2 | — | |
CIUXWRBSDIAJKR
|
6.3 | IC50 | 3 | Yes | |
LVEQCWIYSFCXHR
|
6.3 | IC50 | 3 | — | |
PUIQBGZLGGGFGO
|
6.3 | IC50 | 2 | — | |
BECWPNYJZIVGFM
|
6.3 | IC50 | 3 | Yes | |
BXNRVJLIEMQDOL
|
6.3 | IC50 | 3 | — | |
BYWFNZWJIKYEJQ
|
6.3 | IC50 | 3 | Yes | |
IJCDWDJDJPZXSX
|
6.3 | IC50 | 5 | — | |
RMXCVAFRLLKAJD
|
6.3 | IC50 | 3 | Yes | |
UJRBNGYJDIGSOL
|
6.3 | IC50 | 5 | — | |
CKADUCCMLBGQGD
|
6.3 | IC50 | 3 | Yes | |
KLGPIUGVYNHCJD
|
6.3 | IC50 | 3 | Yes | |
ROYSOBXGDVHDTQ
|
6.3 | IC50 | 5 | Yes | |
RHJUQZKMGKSJEL
|
6.3 | IC50 | 3 | — | |
JHPYFDJWXXWGRB
|
6.2 | IC50 | 3 | Yes | |
RSBDIBAMWNTGCI
|
6.2 | IC50 | 2 | — | |
UUVHQULSIKGMES
|
6.2 | IC50 | 2 | — | |
YFMNOAQQYQDPRP
|
6.2 | IC50 | 3 | — | |
DJYOAYPWIWACRH
|
6.2 | IC50 | 3 | Yes | |
SVHNBCYOOFGBDY
|
6.2 | IC50 | 3 | — | |
WAHQJJLIQLLJGD
|
6.2 | IC50 | 3 | Yes | |
WJLNAPDUWBBQHL
|
6.2 | IC50 | 3 | Yes | |
NZQKBSXOPCGJGL
|
6.2 | IC50 | 3 | — | |
XHIISTKHRQWJJN
|
6.2 | IC50 | 3 | Yes | |
IVHZRYBZVXHBJC
|
6.2 | IC50 | 3 | Yes |