Target Details
| UniProt AC | P53609 |
|---|---|
| Gene Symbol | PGGT1B |
| Protein Name | Geranylgeranyl transferase type-1 subunit beta |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00432 (Prenyltrans) |
Summary
- Multi-target molecules 232
- Clinical molecules 172
- Avg pChEMBL 7.05
Active Molecules (232)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YGJHSCAJBDJRFY
|
7.0 | IC50 | 3 | Yes | |
AYVGITDSDRJQKI
|
7.0 | IC50 | 3 | Yes | |
DRDJJFGPXROAMP
|
7.0 | IC50 | 3 | Yes | |
JNUGFGAVPBYSHF
|
7.0 | IC50 | 5 | Yes | |
OINNEUNVOZHBOX
|
7.0 | IC50 | 2 | — | |
AEUOJCZWQRBEMN
|
7.0 | IC50 | 3 | Yes | |
HQQOMOWVWPBVRR
|
7.0 | IC50 | 3 | Yes | |
PIHDHMFGLZPELL
|
7.0 | IC50 | 2 | — | |
WUBHEKLVWNZHSF
|
7.0 | IC50 | 3 | Yes | |
ZAUBGERWKXAZHI
|
7.0 | IC50 | 3 | Yes | |
JQBMSMWRNHYILW
|
6.9 | IC50 | 3 | Yes | |
MQBSRXJKDKCOAM
|
6.9 | IC50 | 3 | Yes | |
CQCNIBNGGPUKMH
|
6.9 | IC50 | 3 | Yes | |
WHPKJYJVLZBIAP
|
6.9 | IC50 | 3 | Yes | |
BPPQKJVLUWXNRM
|
6.9 | IC50 | 4 | Yes | |
DISVQWQQQWMFSB
|
6.8 | IC50 | 2 | — | |
IDCVPCYUIWJZSF
|
6.8 | IC50 | 2 | — | |
IDVLFUHLBYSGQS
|
6.8 | IC50 | 3 | Yes | |
CPUPJBLXXHGNPV
|
6.8 | IC50 | 2 | Yes | |
DWFPFAQHVZRKBX
|
6.8 | IC50 | 3 | Yes | |
ITOOXSJDSBTQNY
|
6.8 | IC50 | 3 | Yes | |
MNUNZZHRDOMTJY
|
6.8 | IC50 | 3 | Yes | |
QCKHJKGNCCPADL
|
6.8 | IC50 | 2 | — | |
RBZQXEMPWMGPEK
|
6.8 | IC50 | 3 | — | |
SUTIPWLBYIUOBW
|
6.8 | IC50 | 3 | Yes | |
VRUYMJKZIKNSKH
|
6.8 | IC50 | 3 | Yes | |
XVWPFYDMUFBHBF
|
6.8 | IC50 | 2 | — | |
HBYRYAHMXSFRDA
|
6.8 | IC50 | 2 | Yes | |
AQTMMHDZTUQGJD
|
6.8 | IC50 | 3 | Yes | |
NIKJJDARCUJOSC
|
6.8 | IC50 | 3 | Yes | |
HCTZGNQLYBGGPK
|
6.8 | IC50 | 2 | — | |
FISVBHHSQNPBPG
|
6.8 | IC50 | 3 | Yes | |
NKNMRYCDVOOEKZ
|
6.7 | IC50 | 3 | Yes | |
BLEVYVOQEISZIT
|
6.7 | IC50 | 3 | Yes | |
VSJRZQRFGNBQRA
|
6.7 | IC50 | 2 | — | |
VSJRZQRFGNBQRA
|
6.7 | IC50 | 3 | Yes | |
DUORQQSLNAGSSQ
|
6.7 | IC50 | 3 | Yes | |
WKLYKVGIWYWSHH
|
6.7 | IC50 | 2 | Yes | |
YRURVXAIOAEGME
|
6.7 | IC50 | 2 | — | |
QKFHVTMTAUFWNT
|
6.7 | IC50 | 3 | Yes | |
PTNBPPZVBINDKZ
|
6.7 | IC50 | 3 | Yes | |
ZEIRRWOZIKZYIO
|
6.7 | IC50 | 3 | Yes | |
RDECPKAPXFKZRQ
|
6.6 | IC50 | 3 | Yes | |
HPODVVZGZWGVDV
|
6.6 | IC50 | 2 | — | |
MFPPMKRAKTUYMX
|
6.6 | IC50 | 3 | Yes | |
TXMWWHNPHYEWNP
|
6.6 | IC50 | 3 | Yes | |
XOFBXIHLMNJMOE
|
6.6 | IC50 | 3 | Yes | |
CMGIYMUBWMWULU
|
6.6 | IC50 | 2 | — | |
JERRNUSBLOXSHR
|
6.6 | IC50 | 2 | Yes | |
AQAZIJJBKQIIAP
|
6.5 | IC50 | 3 | Yes |