Target Details
| UniProt AC | P53609 |
|---|---|
| Gene Symbol | PGGT1B |
| Protein Name | Geranylgeranyl transferase type-1 subunit beta |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00432 (Prenyltrans) |
Summary
- Multi-target molecules 232
- Clinical molecules 172
- Avg pChEMBL 7.05
Active Molecules (232)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZBRVJLSHNVWEKS
|
7.8 | IC50 | 3 | Yes | |
VSZXKSCVZMOQFB
|
7.7 | IC50 | 3 | Yes | |
VKLQBYODSYOXOK
|
7.7 | IC50 | 3 | Yes | |
YIHOJJQZGPJKGV
|
7.7 | IC50 | 3 | Yes | |
GAJLKAVQYXFCRU
|
7.7 | IC50 | 2 | — | |
FZJOMPQKENNHGD
|
7.7 | IC50 | 3 | Yes | |
JRTOBKVVIBBEQD
|
7.6 | IC50 | 2 | Yes | |
ACXPVQQIYOUAGF
|
7.6 | IC50 | 3 | Yes | |
KMNYYAJYASNHCC
|
7.6 | IC50 | 3 | — | |
BVCQRIMNJALALQ
|
7.5 | IC50 | 3 | Yes | |
QGCNWBQUPNGUPL
|
7.5 | IC50 | 3 | Yes | |
IGCORMDACWRGMB
|
7.5 | IC50 | 3 | Yes | |
LIRHXIGWHONJAQ
|
7.5 | IC50 | 3 | Yes | |
WWBMVHKTRROALT
|
7.5 | IC50 | 2 | — | |
CNHFDLPFXKHRKU
|
7.5 | IC50 | 3 | Yes | |
WLEUBRYSZJGDFY
|
7.5 | IC50 | 3 | — | |
ODTFPKNIFYMEHP
|
7.4 | IC50 | 2 | Yes | |
WLEUBRYSZJGDFY
|
7.4 | IC50 | 4 | — | |
NAEYWVZYJOIXPA
|
7.4 | IC50 | 3 | Yes | |
YOSWFXLZVOUMIC
|
7.4 | IC50 | 3 | Yes | |
LQNDTMZXYCNVNE
|
7.4 | IC50 | 2 | Yes | |
ABMQIHFTAMGDJE
|
7.3 | IC50 | 3 | Yes | |
NMPOEHMYTSFAOT
|
7.3 | IC50 | 3 | Yes | |
DBWZOKRHHKZPJP
|
7.3 | IC50 | 3 | — | |
DJVTZQIKKLGURV
|
7.3 | IC50 | 3 | Yes | |
RZBRPHGLFWWUEG
|
7.3 | IC50 | 3 | Yes | |
ZIXDDEATQSBHHL
|
7.3 | IC50 | 5 | Yes | |
PKMVDYSKPDHRLR
|
7.3 | IC50 | 3 | Yes | |
MHNMEERHZSPWFL
|
7.3 | IC50 | 3 | — | |
XVWPFYDMUFBHBF
|
7.3 | IC50 | 2 | — | |
IZYCQMKDUPSJSI
|
7.3 | IC50 | 3 | Yes | |
PHGAACKWQSAJHR
|
7.2 | IC50 | 2 | Yes | |
QAIUZYFKQAGOBZ
|
7.2 | IC50 | 3 | Yes | |
RAWVEDVPUJQLEN
|
7.2 | IC50 | 2 | Yes | |
LONOBJYLFFURAI
|
7.2 | IC50 | 3 | Yes | |
ZJVHZEHEHYNPCV
|
7.2 | IC50 | 2 | Yes | |
MJSIQIQTEIQMNA
|
7.2 | IC50 | 2 | — | |
YUFXAWQITMCWMO
|
7.1 | IC50 | 3 | Yes | |
VTPCNRSHUJQADS
|
7.1 | IC50 | 3 | Yes | |
ODNODBYULJCPOM
|
7.1 | IC50 | 3 | Yes | |
LUQBIRLUHCYXQM
|
7.1 | IC50 | 3 | Yes | |
PPSUJYUXOZCAFU
|
7.1 | IC50 | 3 | Yes | |
HGDNILFTURGNIL
|
7.1 | IC50 | 3 | Yes | |
FJGNOYWWYBUMAR
|
7.0 | IC50 | 2 | — | |
KZMSAVPDHMHSQO
|
7.0 | IC50 | 2 | Yes | |
QMBOMETUAPMBFM
|
7.0 | IC50 | 3 | Yes | |
DXJRWWRZZPRGJB
|
7.0 | IC50 | 3 | Yes | |
ZPHPMNJCCXXCGX
|
7.0 | IC50 | 3 | Yes | |
QFVRKKGXFGGVET
|
7.0 | IC50 | 3 | Yes | |
RBZQXEMPWMGPEK
|
7.0 | IC50 | 3 | — |