Target Details
| UniProt AC | P53609 |
|---|---|
| Gene Symbol | PGGT1B |
| Protein Name | Geranylgeranyl transferase type-1 subunit beta |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00432 (Prenyltrans) |
Summary
- Multi-target molecules 232
- Clinical molecules 172
- Avg pChEMBL 7.05
Active Molecules (232)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WARZQQRPINBDAJ
|
9.8 | IC50 | 3 | Yes | |
VQNYIQPZXRNJMG
|
9.7 | IC50 | 3 | Yes | |
QGPSHWUWMGSFJB
|
9.5 | IC50 | 3 | Yes | |
QOTXVDPQOVHXPX
|
9.5 | IC50 | 3 | Yes | |
XRJFAINHZHMKOK
|
9.2 | IC50 | 3 | Yes | |
KVTUJRZUQCULNT
|
9.1 | IC50 | 3 | Yes | |
SHUCBLWUZXSRAC
|
9.1 | IC50 | 3 | Yes | |
YDQQLXXIRZYPPK
|
8.9 | IC50 | 3 | Yes | |
WKHUKTIZMOPZJE
|
8.8 | IC50 | 3 | Yes | |
YIZSZHVXFHAUCR
|
8.8 | IC50 | 3 | Yes | |
FUMOSLFZEUUPBJ
|
8.7 | IC50 | 3 | Yes | |
XUQVGNQCLMEBOL
|
8.7 | IC50 | 3 | Yes | |
OFEALQXVDCUNBG
|
8.6 | IC50 | 3 | Yes | |
CPCCCCDBCSOFNS
|
8.6 | IC50 | 3 | Yes | |
QRWYVPGOSHKJPP
|
8.5 | IC50 | 3 | Yes | |
GTURWVWPNOUBNH
|
8.5 | IC50 | 3 | Yes | |
MHNMEERHZSPWFL
|
8.4 | IC50 | 3 | Yes | |
MHNMEERHZSPWFL
|
8.3 | IC50 | 3 | — | |
ASUWZCFQGVUVGX
|
8.3 | IC50 | 3 | Yes | |
HZUKRNKCJCVHQD
|
8.3 | IC50 | 2 | — | |
LMXZFNUEMHAYLD
|
8.3 | IC50 | 3 | Yes | |
IIPCWBJMJZVLOK
|
8.3 | IC50 | 3 | — | |
QMCCVNYWKLFKCQ
|
8.3 | IC50 | 2 | — | |
MHNMEERHZSPWFL
|
8.3 | IC50 | 3 | Yes | |
KMNYYAJYASNHCC
|
8.2 | IC50 | 3 | Yes | |
ARBOPWPZIKDYTB
|
8.1 | IC50 | 2 | — | |
IENQPUVVSDIXCT
|
8.1 | IC50 | 3 | Yes | |
KMNYYAJYASNHCC
|
8.1 | IC50 | 3 | Yes | |
HKGUHEGKBLYKHY
|
8.1 | Ki | 3 | Yes | |
ZFBGYVVVVKZTFW
|
8.1 | IC50 | 3 | Yes | |
QRZPLNXYFZWRNQ
|
8.1 | IC50 | 3 | Yes | |
RPSVZMJVPOGOLG
|
8.1 | IC50 | 3 | Yes | |
XWUNACODWZDLMP
|
8.0 | IC50 | 3 | Yes | |
COLCNDRDBCLVOC
|
8.0 | IC50 | 2 | — | |
RHTSWGZKPCQUKZ
|
8.0 | IC50 | 3 | Yes | |
DOZZPCQVJJBKME
|
8.0 | IC50 | 3 | Yes | |
GEOWAWJUOWQWJH
|
8.0 | IC50 | 3 | Yes | |
GOYDJMAPJITTBZ
|
8.0 | IC50 | 2 | — | |
ZORLZQLLRSELQH
|
8.0 | IC50 | 2 | Yes | |
BMGIODYUKGDYTO
|
7.9 | IC50 | 3 | Yes | |
MHNMEERHZSPWFL
|
7.9 | IC50 | 3 | — | |
ZCCICPFBBPENMT
|
7.9 | IC50 | 3 | Yes | |
OBXLXUGOZZWQOW
|
7.9 | IC50 | 4 | Yes | |
SHPJZFRGYYTFJF
|
7.8 | IC50 | 3 | Yes | |
DSUYZKFAJRJFFP
|
7.8 | IC50 | 2 | — | |
OAEIWTGUZXTPAT
|
7.8 | IC50 | 3 | Yes | |
QAQOQARNGPJYIW
|
7.8 | IC50 | 2 | — | |
ULZTVJKTSYZRPI
|
7.8 | IC50 | 2 | — | |
UUNGZSLCFUPOGA
|
7.8 | IC50 | 3 | Yes | |
PMCYJSRQOFQRLF
|
7.8 | IC50 | 3 | Yes |