Target Details
| UniProt AC | P53582 |
|---|---|
| Gene Symbol | METAP1 |
| Protein Name | Methionine aminopeptidase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00557 (Peptidase_M24) PF15801 (zf-C6H2) |
Summary
- Multi-target molecules 5
- Clinical molecules 0
- Avg pChEMBL 6.23
Active Molecules (5)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AIIOXZPEXXZCML
|
6.4 | IC50 | 2 | — | |
QBMYJIFXSXKPFS
|
6.4 | IC50 | 2 | — | |
NKASPYGDXVCCTA
|
6.2 | IC50 | 2 | — | |
XSYJUVKQRPLTAU
|
6.2 | IC50 | 2 | — | |
DZZIDDGXTTVGSU
|
6.0 | IC50 | 2 | — |