Target Details
| UniProt AC | P53355 |
|---|---|
| Gene Symbol | DAPK1 |
| Protein Name | Death-associated protein kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00023 (Ank) PF12796 (Ank_2) PF13637 (Ank_4) PF00531 (Death) PF00069 (Pkinase) |
Summary
- Multi-target molecules 37
- Clinical molecules 4
- Avg pChEMBL 6.83
KEGG Pathways (3)
Associated Diseases (1)
Active Molecules (37)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKSZLNNOFSGOKW
|
8.8 | Kd | 213 | — | |
LYADGAGFYYXXIO
|
8.7 | IC50 | 82 | — | |
HKSZLNNOFSGOKW
|
8.0 | IC50 | 408 | — | |
YMZURUFTCLYPGO
|
7.9 | IC50 | 4 | — | |
JOOXLOJCABQBSG
|
7.8 | Kd | 139 | — | |
LOONVQWRKJLEEG
|
7.6 | IC50 | 8 | — | |
NGFGTMFVWSDFPS
|
7.6 | IC50 | 32 | — | |
MJWLCXWVFUXXNZ
|
7.3 | Kd | 3 | — | |
NHHQJBCNYHBUSI
|
7.3 | Kd | 220 | — | |
OSVUGUHRKMMBSE
|
7.2 | Kd | 170 | — | |
NXSJMRCTGYTSTK
|
7.2 | Kd | 200 | — | |
HFNKQEVNSGCOJV
|
7.1 | Kd | 65 | — | |
UIARLYUEJFELEN
|
7.1 | Kd | 289 | Yes | |
MFAQYJIYDMLAIM
|
7.0 | Kd | 130 | Yes | |
WINHZLLDWRZWRT
|
6.9 | Kd | 201 | Yes | |
YQMFNWQNASFQAE
|
6.8 | IC50 | 5 | — | |
WLKJMISWXHORCR
|
6.7 | IC50 | 11 | — | |
MCIDHQCNUZBVQJ
|
6.6 | IC50 | 2 | — | |
NASYEGAVCTZSDO
|
6.6 | Kd | 5 | — | |
CTNPALGJUAXMMC
|
6.6 | Kd | 151 | — | |
YYLKKYCXAOBSRM
|
6.4 | Kd | 191 | — | |
ZUKXESAZGMJHLJ
|
6.4 | IC50 | 4 | — | |
NXWXUDHOUKWAQU
|
6.4 | Kd | 16 | — | |
MCUJKPPARUPFJM
|
6.4 | Kd | 11 | — | |
LIMMMAWLSIHXGX
|
6.3 | IC50 | 5 | — | |
VVFCWFGNLTVHBL
|
6.3 | IC50 | 5 | — | |
XKQNBVAZAFAZFL
|
6.3 | IC50 | 6 | — | |
XQVVPGYIWAGRNI
|
6.3 | Kd | 34 | — | |
SVNVPNHWFJFRLZ
|
6.2 | IC50 | 8 | — | |
HZTYDQRUAWIZRE
|
6.2 | Kd | 40 | Yes | |
QVJYGMLAIWRCFT
|
6.2 | IC50 | 5 | — | |
RYJMAXSFHOPKJH
|
6.1 | IC50 | 2 | — | |
ZVSNSFQQKSZZMY
|
6.1 | IC50 | 7 | — | |
ZCBUQCWBWNUWSU
|
6.0 | Kd | 59 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |