Target Details
| UniProt AC | P53350 |
|---|---|
| Gene Symbol | PLK1 |
| Protein Name | Serine/threonine-protein kinase PLK1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00659 (POLO_box) |
Summary
- Multi-target molecules 357
- Clinical molecules 33
- Avg pChEMBL 7.56
KEGG Pathways (4)
Active Molecules (357)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FMCBJKDUHHIOQB
|
6.3 | IC50 | 2 | — | |
HEVBIDCNQYUCRF
|
6.3 | IC50 | 2 | — | |
QAXOLKUTJAQVHO
|
6.3 | IC50 | 3 | — | |
UMJFDLYATACWKW
|
6.3 | IC50 | 2 | — | |
GXNUDSNBBQOPIA
|
6.3 | IC50 | 4 | — | |
AKWNDIGQZONPHP
|
6.3 | IC50 | 2 | — | |
CLEGDJQQHUTCOW
|
6.3 | Ki | 43 | — | |
DVMCRBPTCKGCAX
|
6.3 | IC50 | 2 | — | |
MASJMHFQMYAPJR
|
6.3 | Ki | 41 | — | |
NKGLJTITEFZKAN
|
6.3 | Ki | 35 | — | |
OWDRQHVEJIYVOI
|
6.3 | Ki | 47 | — | |
RJZDECGDCKOHBV
|
6.3 | Ki | 70 | — | |
IGNHIECBXXHFPK
|
6.3 | IC50 | 2 | — | |
VAPOMSIOLKMAIW
|
6.3 | Ki | 7 | — | |
BMCKWRUTJXVUFF
|
6.3 | IC50 | 4 | — | |
BRLRIFFHVZNKFH
|
6.3 | IC50 | 2 | — | |
DTKNQMRYSGVPEX
|
6.3 | IC50 | 3 | — | |
KPXMSUZHJCHOTN
|
6.3 | IC50 | 3 | — | |
LCBAQTCTQXHTJG
|
6.2 | IC50 | 9 | — | |
AILRADAXUVEEIR
|
6.2 | IC50 | 75 | — | |
TZSJMSZEKQGCBI
|
6.2 | Ki | 15 | — | |
DKPUPJUELCIYFX
|
6.2 | IC50 | 2 | — | |
IBUMAHMUIWPTCV
|
6.2 | IC50 | 3 | — | |
JGIBKTCCYJBOMS
|
6.2 | IC50 | 2 | — | |
KHBSTEQSSXYFCY
|
6.2 | IC50 | 2 | — | |
MUOKSQABCJCOPU
|
6.2 | Kd | 36 | — | |
PYVMYBZZIWFCPE
|
6.2 | IC50 | 2 | — | |
QHPKKGUGRGRSGA
|
6.1 | IC50 | 7 | Yes | |
QWAOMERKQXGSJH
|
6.1 | IC50 | 2 | — | |
XFHCCTMTQFFLCT
|
6.1 | IC50 | 2 | — | |
IRDQZYNDOWVJIZ
|
6.1 | IC50 | 2 | — | |
PMMISILPBLQWSZ
|
6.1 | IC50 | 2 | — | |
BQPLWJRDSDNGNE
|
6.1 | Ki | 16 | — | |
GBOOMURPCSMHOP
|
6.1 | IC50 | 2 | — | |
LDTAHRLHGHFHKP
|
6.1 | IC50 | 3 | — | |
MVJMMLFMPWITEJ
|
6.1 | Ki | 110 | — | |
DNZGEPPZYMAFLN
|
6.1 | IC50 | 2 | — | |
NHHQJBCNYHBUSI
|
6.1 | Kd | 220 | — | |
RCMAMGZVMIYCFL
|
6.1 | IC50 | 2 | — | |
GNFVJCMQLYMYRH
|
6.1 | IC50 | 2 | — | |
HJKBVLZABNNRFO
|
6.1 | IC50 | 5 | Yes | |
KRFAHCVCYDZSOI
|
6.0 | IC50 | 2 | — | |
XOZJRQDITIJPCH
|
6.0 | IC50 | 2 | — | |
HHYUCVASUIGARF
|
6.0 | IC50 | 4 | — | |
GHPFSYCYZJKVDZ
|
6.0 | Ki | 18 | Yes | |
JXRYPFSBKNWJBW
|
6.0 | IC50 | 4 | — | |
AORZPRLVKUMTOJ
|
6.0 | IC50 | 2 | — | |
DKXHSOUZPMHNIZ
|
6.0 | IC50 | 51 | Yes | |
AENKGHPUTMOKKU
|
6.0 | IC50 | 2 | — | |
BNLPAUPVSCPTDM
|
6.0 | Ki | 15 | — |