Target Details
| UniProt AC | P53350 |
|---|---|
| Gene Symbol | PLK1 |
| Protein Name | Serine/threonine-protein kinase PLK1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00659 (POLO_box) |
Summary
- Multi-target molecules 357
- Clinical molecules 33
- Avg pChEMBL 7.56
KEGG Pathways (4)
Active Molecules (357)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IRCDNPBWELYZBD
|
6.8 | IC50 | 3 | — | |
CIGSBKXHEYMHAF
|
6.8 | IC50 | 2 | — | |
GCPQQOBOYKBWPO
|
6.8 | IC50 | 2 | — | |
ZJDFSKSBQBPOSK
|
6.8 | IC50 | 24 | Yes | |
HNLPHJIQJRDKKX
|
6.8 | IC50 | 2 | — | |
YYEWDYMBVPPZDJ
|
6.8 | IC50 | 2 | — | |
BNJAETMQKIKKSN
|
6.7 | IC50 | 2 | — | |
XWQNZYCWLMEIBB
|
6.7 | IC50 | 5 | Yes | |
LKUJDAHYLPICSE
|
6.7 | Ki | 24 | — | |
LTQRUCOWRVPXHK
|
6.7 | Kd | 2 | — | |
RKKIDHHGKNGTQI
|
6.7 | Ki | 28 | — | |
UYJNQQDJUOUFQJ
|
6.7 | Ki | 68 | — | |
DAAGOCSHXCDWDY
|
6.7 | IC50 | 3 | — | |
UIARLYUEJFELEN
|
6.7 | Kd | 289 | Yes | |
HKSZLNNOFSGOKW
|
6.7 | IC50 | 408 | — | |
KMZDOKNRRSNTSW
|
6.7 | IC50 | 2 | — | |
MLSIWMLVUIWYLH
|
6.6 | Ki | 2 | — | |
WGZYFFJOGZFXBF
|
6.6 | IC50 | 2 | — | |
ZYQXOZKYXADECC
|
6.6 | IC50 | 5 | Yes | |
FUMCKNCUEAQHCV
|
6.6 | Ki | 103 | — | |
KOKNYBBQIVDZCK
|
6.6 | IC50 | 2 | — | |
NILXCNICWMPUMM
|
6.6 | IC50 | 2 | — | |
UEIRKXUBXCSHJE
|
6.6 | Ki | 19 | — | |
XCYGTFKOOGNUMR
|
6.6 | IC50 | 5 | Yes | |
GEGMKHTYQVNYFV
|
6.6 | IC50 | 2 | — | |
GYDZFEKAOMUPJL
|
6.6 | IC50 | 2 | — | |
FRVAEEMWIWELKQ
|
6.5 | IC50 | 2 | — | |
JOOXLOJCABQBSG
|
6.5 | Kd | 139 | — | |
ZSYVDZWVCFZJLJ
|
6.5 | IC50 | 2 | — | |
TWABWUVZWXSPTC
|
6.5 | IC50 | 3 | — | |
WPPGBVWZGMDXKF
|
6.5 | IC50 | 5 | — | |
CKVWQORGCCEYHS
|
6.5 | Ki | 50 | — | |
KBRJIBFRLFVYJL
|
6.5 | Ki | 5 | — | |
RHIJMDNVEPLDED
|
6.5 | IC50 | 2 | — | |
YQXSREGMIKNZEU
|
6.5 | Ki | 8 | — | |
OXMBEXXWWXTOCD
|
6.5 | IC50 | 2 | — | |
MKMWADKTKCUOBJ
|
6.5 | IC50 | 2 | — | |
NUQUWKXNHFMEAJ
|
6.5 | IC50 | 3 | — | |
SKCATAJFICHYLV
|
6.5 | IC50 | 2 | — | |
INBHXNZJARFRRF
|
6.5 | IC50 | 2 | — | |
ANAAVHLLZPPWCU
|
6.4 | IC50 | 6 | — | |
RHNQIPARHTZKOF
|
6.4 | IC50 | 2 | — | |
UMJFDLYATACWKW
|
6.4 | IC50 | 2 | — | |
LYNBNVBMAGDJRW
|
6.4 | Ki | 81 | — | |
UVZVWLFSZNPMBS
|
6.4 | Ki | 17 | — | |
VNGYQBMDQMDALH
|
6.4 | Ki | 25 | — | |
OQCYIOKKFGCDSR
|
6.4 | IC50 | 4 | Yes | |
UNVPHVSVVHLLKD
|
6.4 | IC50 | 2 | — | |
URBLFMVEDFWKGZ
|
6.4 | IC50 | 6 | — | |
YQCCDKOFONLPFF
|
6.4 | IC50 | 2 | — |