Target Details
| UniProt AC | P53350 |
|---|---|
| Gene Symbol | PLK1 |
| Protein Name | Serine/threonine-protein kinase PLK1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00659 (POLO_box) |
Summary
- Multi-target molecules 357
- Clinical molecules 33
- Avg pChEMBL 7.56
KEGG Pathways (4)
Active Molecules (357)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QIWKCZYPLMKZJX
|
7.3 | IC50 | 2 | — | |
UXNCNPVLRQGOMH
|
7.3 | IC50 | 3 | — | |
WUDDKNUPJTYVAB
|
7.3 | Kd | 2 | — | |
AHUQZOZSCWOMOS
|
7.3 | IC50 | 4 | — | |
KVJXBCZPOFTDAU
|
7.3 | IC50 | 2 | — | |
IJDPNONZYDDAHT
|
7.3 | IC50 | 3 | — | |
JTYDPPQNZSHIQR
|
7.3 | IC50 | 2 | — | |
UZVJWQPORUUHRW
|
7.3 | IC50 | 3 | — | |
MRITYVDXXFOOAU
|
7.3 | Kd | 6 | — | |
JECZPVPRJJYJME
|
7.2 | IC50 | 2 | — | |
HKERRRNEVQHIRB
|
7.2 | IC50 | 2 | — | |
OAVGBZOFDPFGPJ
|
7.2 | Ki | 42 | Yes | |
OWRXHGAFWZFFCW
|
7.2 | Ki | 113 | — | |
ZBJWJVGFIIULBV
|
7.2 | IC50 | 3 | — | |
XDRHCUWKZRZSEP
|
7.2 | IC50 | 2 | — | |
IJNMRIYHRCSVCO
|
7.2 | IC50 | 3 | — | |
UTHWBIPHRYUJSU
|
7.2 | IC50 | 11 | Yes | |
FRVZZHQYKGFUEH
|
7.2 | IC50 | 2 | — | |
VBYSCQVUJACHHJ
|
7.2 | IC50 | 2 | — | |
NCDFJOWBEBTLBV
|
7.1 | IC50 | 2 | — | |
DYAVJUMLONUWEK
|
7.1 | IC50 | 2 | — | |
JCFJQIHDZHHMQT
|
7.1 | Ki | 42 | — | |
QBQNTNGYPHAFJA
|
7.1 | IC50 | 2 | — | |
LYAOPUXRPJKSKW
|
7.1 | IC50 | 3 | — | |
BIIPWGFUTBPTNQ
|
7.1 | IC50 | 2 | — | |
TWYRQXNMQMYEGC
|
7.0 | IC50 | 2 | — | |
CFTIJALKSHXVNU
|
7.0 | IC50 | 3 | — | |
NMVMZFAZMNUQMX
|
7.0 | IC50 | 2 | — | |
UNZVQIJLQQYQLN
|
7.0 | IC50 | 6 | — | |
DTEKTGDVSARYDS
|
7.0 | IC50 | 11 | — | |
OMOOZNJIAYMBSP
|
7.0 | IC50 | 5 | Yes | |
MMGBSWRVNVBEIM
|
7.0 | IC50 | 2 | — | |
NQROQCRXQDNZSD
|
7.0 | IC50 | 3 | — | |
QXAKKDDDYAESLJ
|
7.0 | IC50 | 6 | Yes | |
YOMURATVIWHSOR
|
7.0 | IC50 | 2 | — | |
ZOBRPBVIEUWYJR
|
7.0 | IC50 | 5 | Yes | |
GCFCQBCBKXQUCD
|
6.9 | IC50 | 3 | — | |
MCJYLZXJWVLMLI
|
6.9 | IC50 | 2 | — | |
HTPNGOWITIWAHM
|
6.9 | IC50 | 3 | — | |
OYDGHJTZNAFKAQ
|
6.9 | IC50 | 6 | Yes | |
QYUSWNWUSZFQJV
|
6.9 | IC50 | 2 | — | |
HFNKQEVNSGCOJV
|
6.9 | Kd | 65 | — | |
WPIFRGDKXSWKPX
|
6.9 | IC50 | 5 | Yes | |
YZOJFEPZEVKWPV
|
6.9 | IC50 | 2 | — | |
YTJXTZVLUBWOAJ
|
6.8 | IC50 | 2 | — | |
UUINGAOFFFDPBY
|
6.8 | IC50 | 5 | Yes | |
DPROZSHCTFNYSW
|
6.8 | IC50 | 6 | Yes | |
OGBRMNPYWOVJQQ
|
6.8 | IC50 | 2 | — | |
DHMVFGZTRVZQFI
|
6.8 | IC50 | 2 | — | |
GCBJDOWIQHMCMR
|
6.8 | Ki | 84 | — |