Target Details
| UniProt AC | P53350 |
|---|---|
| Gene Symbol | PLK1 |
| Protein Name | Serine/threonine-protein kinase PLK1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00659 (POLO_box) |
Summary
- Multi-target molecules 357
- Clinical molecules 33
- Avg pChEMBL 7.56
KEGG Pathways (4)
Active Molecules (357)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PRMNYSLMFFRETJ
|
7.8 | IC50 | 3 | — | |
PVVRSMIEEGPASF
|
7.8 | IC50 | 3 | — | |
VZLKEAGJBNAJKB
|
7.8 | IC50 | 2 | — | |
YXRJOXHIGGNCBU
|
7.8 | IC50 | 3 | — | |
SONVWPLFNTVESG
|
7.8 | IC50 | 12 | — | |
NERSFQYNEXMEPK
|
7.7 | IC50 | 3 | — | |
VJDBYVPTQWPRPA
|
7.7 | Kd | 2 | — | |
KBILTEUAXWLXKP
|
7.7 | Kd | 2 | — | |
NMIWWLZKGDETAG
|
7.7 | IC50 | 2 | — | |
NCCZKHZUPCPIOT
|
7.7 | IC50 | 3 | — | |
QQWUGDVOUVUTOY
|
7.7 | Kd | 231 | Yes | |
AUWBCLDCSRIWGM
|
7.7 | IC50 | 12 | — | |
AILANCLYZDKELS
|
7.7 | IC50 | 3 | — | |
MVOGKCYGDBWOLZ
|
7.7 | IC50 | 2 | — | |
QLUYMIVVAYRECT
|
7.7 | Kd | 12 | — | |
RNCCSJOQZGLCIQ
|
7.7 | IC50 | 3 | — | |
VBDIOKSSYUZONA
|
7.7 | IC50 | 3 | — | |
ZDQJNYLFGPXANH
|
7.7 | IC50 | 3 | — | |
QUMCIHKVKQYNPA
|
7.7 | IC50 | 2 | — | |
UEILKDPTXUZCFH
|
7.6 | IC50 | 3 | — | |
XWNHXTVCPNRSTM
|
7.6 | IC50 | 3 | — | |
ITDUQSWFIDASGI
|
7.6 | IC50 | 3 | — | |
MLSKNMPNUOPUAB
|
7.6 | IC50 | 3 | — | |
ZHZUHNWBNIKEGE
|
7.5 | IC50 | 2 | — | |
FGUYNCHKIOFPMS
|
7.5 | IC50 | 2 | — | |
NMIWWLZKGDETAG
|
7.5 | IC50 | 2 | — | |
QIMUQYHRHHNTNY
|
7.5 | IC50 | 3 | — | |
QMAVWDJUBQEBDQ
|
7.5 | IC50 | 2 | — | |
UHCHLTQBLNUYRT
|
7.5 | IC50 | 2 | — | |
SQRHNUCMJHZAKJ
|
7.5 | IC50 | 2 | — | |
YMIJUBCSOKSFRU
|
7.5 | Ki | 87 | — | |
GSXMJWLLQORXFR
|
7.5 | IC50 | 3 | — | |
LXQFQJQZJHRTKK
|
7.5 | IC50 | 2 | — | |
ITAJXWHXKVYGCF
|
7.5 | IC50 | 5 | — | |
KSMYGTHXVJXRTI
|
7.5 | IC50 | 3 | — | |
RJERVODZSCACGJ
|
7.5 | IC50 | 3 | — | |
SFNMDOXBLCGZMQ
|
7.5 | IC50 | 3 | — | |
LDFXILCAFQHTNH
|
7.4 | IC50 | 3 | — | |
WQQABBZFVHSXMU
|
7.4 | IC50 | 3 | — | |
PKEGAIRYQRMJBD
|
7.4 | IC50 | 2 | — | |
CXPHUBRUHJPONW
|
7.4 | IC50 | 3 | — | |
HOOQLZPFGONGJY
|
7.4 | IC50 | 3 | — | |
HTPNGOWITIWAHM
|
7.4 | IC50 | 3 | — | |
JETXRGKNZYUPEF
|
7.4 | IC50 | 6 | — | |
NTVFVNYEAMJGDF
|
7.4 | IC50 | 3 | — | |
XEXSGNRGTBSSOU
|
7.4 | IC50 | 3 | — | |
XEMJTISGDXHELX
|
7.4 | IC50 | 8 | Yes | |
VMFNGGJHVCGNJO
|
7.4 | IC50 | 2 | — | |
YRUKXDLUMKDTLG
|
7.4 | IC50 | 2 | — | |
HZTYDQRUAWIZRE
|
7.3 | Kd | 40 | Yes |