Target Details
| UniProt AC | P53350 |
|---|---|
| Gene Symbol | PLK1 |
| Protein Name | Serine/threonine-protein kinase PLK1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00659 (POLO_box) |
Summary
- Multi-target molecules 357
- Clinical molecules 33
- Avg pChEMBL 7.56
KEGG Pathways (4)
Active Molecules (357)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BLOOVKYIUMFKLC
|
8.3 | IC50 | 2 | — | |
NHKAFPBCWTVDHF
|
8.3 | IC50 | 2 | — | |
MAULBJVKJOGNGD
|
8.2 | IC50 | 3 | — | |
OCYISXRMEJNANP
|
8.2 | IC50 | 3 | — | |
RCDQFASKGQECOZ
|
8.2 | Ki | 2 | — | |
JYYQJHRWOKIHGC
|
8.2 | IC50 | 3 | — | |
GDMBPOYBSJXINX
|
8.2 | IC50 | 2 | — | |
HWASNOYCCGHVQF
|
8.2 | IC50 | 5 | Yes | |
IBHXQUPAKHOLCH
|
8.2 | IC50 | 2 | — | |
ITYGFIRONBGARW
|
8.2 | IC50 | 3 | — | |
RZFGZSWFNYQBMG
|
8.2 | Ki | 2 | — | |
INCAIRNHZBEWOA
|
8.2 | IC50 | 5 | Yes | |
OPJOIUDMJCRLNO
|
8.2 | IC50 | 2 | — | |
OSCRFGZIFNWYIZ
|
8.1 | IC50 | 3 | — | |
UBHSIXJDGMNJFU
|
8.1 | IC50 | 2 | — | |
VZDOSGQBGHVVCU
|
8.1 | IC50 | 3 | — | |
ZANSQRVTKCXEOP
|
8.1 | IC50 | 2 | — | |
JMDRAMDTWLAOHD
|
8.1 | IC50 | 2 | — | |
QPTZMGCTRHKKJD
|
8.1 | Ki | 3 | — | |
VINNOSMQDSWDTC
|
8.1 | IC50 | 3 | — | |
LBXYVUXGPFEVSI
|
8.1 | IC50 | 3 | — | |
IRXGEPQYGSUCML
|
8.1 | IC50 | 3 | — | |
NXQOLMGRMCDKAS
|
8.1 | IC50 | 2 | — | |
DFHYGDMTHXOWJZ
|
8.1 | IC50 | 2 | — | |
DYQPKOGFUIEBMS
|
8.1 | IC50 | 3 | — | |
JSOGYNPOXPTXNN
|
8.1 | IC50 | 2 | — | |
NLLBMFZASOCLIF
|
8.1 | IC50 | 2 | — | |
OWBFCJROIKNMGD
|
8.1 | IC50 | 3 | — | |
YGQSAYAQCWLSAL
|
8.1 | IC50 | 3 | — | |
FVLMDPWEHBGZDD
|
8.0 | IC50 | 3 | — | |
JKZKKHVTLCFCGS
|
8.0 | IC50 | 3 | — | |
JPWPZFYYVIFSAZ
|
8.0 | IC50 | 3 | — | |
CAVRDKDHKZOOIF
|
8.0 | IC50 | 3 | — | |
FTVMYIRRFFYFIH
|
8.0 | IC50 | 3 | — | |
JQRWYCWILFBHJT
|
8.0 | IC50 | 7 | Yes | |
MIKAKZKNMYZLDX
|
8.0 | Ki | 42 | — | |
QMGCOLHGTKYVOP
|
8.0 | IC50 | 3 | — | |
WCMQEPUDHFATFM
|
8.0 | IC50 | 3 | — | |
MCDYUDVJKXYKNA
|
8.0 | IC50 | 2 | — | |
HJVLRYLCWZPLEP
|
8.0 | IC50 | 2 | — | |
RKWOVOVDWBRGQO
|
8.0 | Kd | 5 | — | |
QDLHCMPXEPAAMD
|
7.9 | IC50 | 13 | Yes | |
DBBQRLYYNNWGPM
|
7.9 | IC50 | 3 | — | |
FLEAYYMORDPWAJ
|
7.9 | Ki | 90 | — | |
TVENGSGQLJMALI
|
7.9 | Ki | 2 | — | |
XANXBCMPWPUNSZ
|
7.9 | IC50 | 3 | — | |
KPDOBADQSPMGFP
|
7.8 | IC50 | 3 | — | |
OXPLZKSKLWBEIM
|
7.8 | IC50 | 8 | Yes | |
ITVQDQHPDYLMCH
|
7.8 | IC50 | 2 | — | |
PGHXJQMSVOKZRE
|
7.8 | IC50 | 3 | — |