Target Details
| UniProt AC | P53350 |
|---|---|
| Gene Symbol | PLK1 |
| Protein Name | Serine/threonine-protein kinase PLK1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00659 (POLO_box) |
Summary
- Multi-target molecules 357
- Clinical molecules 33
- Avg pChEMBL 7.56
KEGG Pathways (4)
Active Molecules (357)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DYQPKOGFUIEBMS
|
9.0 | IC50 | 3 | — | |
NHRDZMBJEDCSLY
|
8.9 | IC50 | 2 | — | |
KZQUEDZXRXCNKM
|
8.9 | IC50 | 2 | — | |
VEUMTIQGKUVYJM
|
8.8 | IC50 | 2 | — | |
CVPAFJFHWHMNPA
|
8.7 | IC50 | 2 | — | |
GILNGUYOGYOZMP
|
8.7 | IC50 | 6 | — | |
IAIOBCSUUBVREO
|
8.7 | IC50 | 8 | Yes | |
IBAYIPZJRQHHLX
|
8.7 | IC50 | 2 | — | |
JAMDNXUAYUHJLJ
|
8.7 | IC50 | 40 | — | |
MYVQSDVXBZNNLF
|
8.7 | IC50 | 8 | Yes | |
NYYQMOVTQNHDLM
|
8.7 | IC50 | 4 | — | |
SWIVJTVGOIXUKC
|
8.7 | IC50 | 9 | — | |
WAMWLVAINQIUBS
|
8.7 | IC50 | 3 | — | |
WRWFZZDBIJLBIJ
|
8.7 | IC50 | 2 | — | |
YIJGUCDNKKHCPF
|
8.7 | IC50 | 2 | — | |
YPKNIQOOBNDEBF
|
8.7 | IC50 | 2 | — | |
GGVHAVDTMKMLJT
|
8.7 | IC50 | 2 | — | |
JSKUWFIZUALZLX
|
8.7 | IC50 | 33 | — | |
ZHJGWYRLJUCMRT
|
8.7 | Ki | 18 | — | |
CVLJBLIMHPEZJC
|
8.5 | IC50 | 2 | — | |
HLHNFPFYQRRGPP
|
8.5 | IC50 | 2 | — | |
MQTVRTKADRPRCF
|
8.5 | IC50 | 2 | — | |
OWRZQDDNDUUITK
|
8.5 | IC50 | 3 | — | |
RTYHQIZCRYJKBV
|
8.5 | IC50 | 3 | — | |
SLGRRBVHGIPHNQ
|
8.5 | IC50 | 2 | — | |
VVQWZQWJWMTPJY
|
8.5 | IC50 | 2 | — | |
VVQWZQWJWMTPJY
|
8.5 | IC50 | 2 | — | |
ZRGJZUSQJGUWJC
|
8.5 | IC50 | 2 | — | |
HYADALKUILXFKH
|
8.5 | IC50 | 2 | — | |
LQPBRMWKFJKVSW
|
8.5 | IC50 | 2 | — | |
AAWUJXDNCDOXTN
|
8.4 | IC50 | 3 | — | |
HYBJJIWZOKSTHG
|
8.4 | IC50 | 2 | — | |
XQVVPGYIWAGRNI
|
8.4 | IC50 | 2 | — | |
OSCRFGZIFNWYIZ
|
8.4 | IC50 | 3 | — | |
DJNZZLZKAXGMMC
|
8.4 | IC50 | 3 | — | |
HLHNFPFYQRRGPP
|
8.4 | IC50 | 2 | — | |
IHOWKSDIGLFLPH
|
8.4 | IC50 | 5 | Yes | |
LCZUOXPDOGJHTF
|
8.4 | IC50 | 2 | — | |
MOSNATYSIYEVTF
|
8.4 | IC50 | 2 | — | |
UMRCTLFOWLGNGP
|
8.4 | IC50 | 2 | — | |
FHOHNZUUIVYNKQ
|
8.4 | IC50 | 2 | — | |
ZAJAQZFUONWQPQ
|
8.4 | IC50 | 3 | — | |
DFKJNGVBNCASDM
|
8.3 | IC50 | 2 | — | |
AJJBWPRLFOMJCY
|
8.3 | IC50 | 3 | — | |
HWIAWKKIXLIVDB
|
8.3 | IC50 | 2 | — | |
MOIBHLHUAXJLCW
|
8.3 | IC50 | 5 | — | |
NDIUYMHNCUTVGE
|
8.3 | Ki | 25 | — | |
QUFVOKRHVJFMNM
|
8.3 | IC50 | 8 | Yes | |
XAEATFZFGRMBDN
|
8.3 | IC50 | 2 | — | |
MVYFNZROIDKPOZ
|
8.3 | IC50 | 3 | — |