Target Details
| UniProt AC | P53350 |
|---|---|
| Gene Symbol | PLK1 |
| Protein Name | Serine/threonine-protein kinase PLK1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00659 (POLO_box) |
Summary
- Multi-target molecules 357
- Clinical molecules 33
- Avg pChEMBL 7.56
KEGG Pathways (4)
Active Molecules (357)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JSZIMXVEMYQOJI
|
9.8 | IC50 | 2 | — | |
FPKFEJQELSGORT
|
9.7 | IC50 | 2 | — | |
LBAXGISUFHVKPW
|
9.5 | IC50 | 2 | — | |
OSBPICGFSLCYPI
|
9.5 | IC50 | 2 | — | |
RUHXXMHOKIHJKY
|
9.5 | IC50 | 2 | — | |
YCNMRNSZEJLPCH
|
9.5 | IC50 | 2 | — | |
XSTRJMHOLBBWNN
|
9.5 | IC50 | 4 | — | |
FBULVHVJQISAMG
|
9.4 | IC50 | 2 | — | |
YXXGXTGIMJQZFA
|
9.4 | IC50 | 2 | — | |
INSOERIUGCDMID
|
9.4 | IC50 | 2 | — | |
CQQFCBITQKNHPX
|
9.3 | IC50 | 4 | — | |
BEILSCWVGFIDJL
|
9.3 | IC50 | 2 | — | |
BQOVFHDJHUGBES
|
9.3 | IC50 | 2 | — | |
HHZMJLZHVLBSKE
|
9.3 | IC50 | 2 | — | |
QKXLHLCDBNXSBT
|
9.3 | IC50 | 2 | — | |
BECCYBZVBSCVDH
|
9.3 | IC50 | 2 | — | |
DQDVRWIYUXKYQR
|
9.3 | IC50 | 2 | — | |
PTCKKLKSUNCGCE
|
9.3 | Ki | 2 | — | |
GVQYCXUWKTZCKO
|
9.2 | IC50 | 2 | — | |
DWDZLNLDCMCRMS
|
9.2 | IC50 | 2 | — | |
FRIZQAUPYMDOBS
|
9.2 | IC50 | 2 | — | |
PIFGWPSMJFVPFI
|
9.1 | IC50 | 2 | — | |
UHCHLTQBLNUYRT
|
9.1 | IC50 | 2 | — | |
OTKIKJDBYKBEOE
|
9.1 | Ki | 3 | — | |
XQVVPGYIWAGRNI
|
9.1 | IC50 | 34 | — | |
SXNJFOWDRLKDSF
|
9.1 | IC50 | 3 | — | |
SXNJFOWDRLKDSF
|
9.1 | IC50 | 8 | — | |
COKMLSIYYSUCIR
|
9.1 | IC50 | 2 | — | |
KHVSTZSCKUIMFH
|
9.0 | Ki | 3 | — | |
ACASXOCRQAMKNU
|
9.0 | IC50 | 2 | — | |
AAVMTXYKUJWQBU
|
9.0 | IC50 | 8 | Yes | |
ABXJJVJJEAFTLI
|
9.0 | IC50 | 4 | — | |
AOYIAMTYZLMCGR
|
9.0 | IC50 | 2 | — | |
ASTXNDZZOAPTNR
|
9.0 | IC50 | 2 | — | |
CXJOVIBONXRCNI
|
9.0 | IC50 | 2 | — | |
DNFIELFWKQLTEZ
|
9.0 | IC50 | 2 | — | |
GGHUWFIXZDQNHR
|
9.0 | IC50 | 8 | Yes | |
JVAPIYLPNKDKAQ
|
9.0 | IC50 | 2 | — | |
KFJDFQDPJGBOJE
|
9.0 | IC50 | 4 | — | |
NXOJBDCDDRAJDO
|
9.0 | IC50 | 3 | — | |
OQIVVQXVRCAEIO
|
9.0 | IC50 | 2 | — | |
OVNJVYZXVSMONK
|
9.0 | IC50 | 3 | — | |
PWEVQXOSGNAHIQ
|
9.0 | IC50 | 2 | — | |
RTDGHNXXZKSIDE
|
9.0 | IC50 | 3 | — | |
RXHOSXWWMGMFAO
|
9.0 | IC50 | 2 | — | |
SVUXDKXAQKMLIM
|
9.0 | IC50 | 2 | — | |
TYQDNFSUWCTPOC
|
9.0 | IC50 | 2 | — | |
WPYKLBCLPYHTFI
|
9.0 | IC50 | 2 | — | |
XWUCTSMJFVUKTR
|
9.0 | IC50 | 2 | — | |
YWNUJKWNTHEOIR
|
9.0 | IC50 | 2 | — |