Target Details
| UniProt AC | P52699 |
|---|---|
| Gene Symbol | N/A |
| Protein Name | Metallo-beta-lactamase IMP-1 |
| Organism | Serratia marcescens |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00753 (Lactamase_B) |
Summary
- Multi-target molecules 1,629
- Clinical molecules 0
- Avg pChEMBL 8.28
Active Molecules (1,629)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LSHYTYHPKFOCBP
|
9.1 | IC50 | 3 | — | |
SHVIQNRXTAJHCL
|
9.1 | IC50 | 4 | — | |
SMMKSMNSJBTZFS
|
9.1 | IC50 | 3 | — | |
VLHWEFRARRJBNF
|
9.1 | IC50 | 3 | — | |
HLEHXKLGZMOEAM
|
9.1 | IC50 | 3 | — | |
JLQLVMLCSVSHON
|
9.1 | IC50 | 4 | — | |
JMROEGRSMUVZFK
|
9.1 | IC50 | 4 | — | |
OTNYOQXNSJHTHV
|
9.1 | IC50 | 3 | — | |
XBPWNORVXZMRHK
|
9.1 | IC50 | 3 | — | |
APZLRISPJJBTHB
|
9.0 | IC50 | 3 | — | |
HHWDWFDDPBTCCL
|
9.0 | IC50 | 3 | — | |
WBCGUARXBURTTF
|
9.0 | IC50 | 3 | — | |
JMGDTOZRWTXGIB
|
9.0 | IC50 | 4 | — | |
JSSNYCYCQLWUEO
|
9.0 | IC50 | 4 | — | |
DGYNHLCPOVDSJN
|
9.0 | IC50 | 3 | — | |
JUCUOMCSSPZOOB
|
9.0 | IC50 | 3 | — | |
MOHHMIRAZDGHTA
|
9.0 | IC50 | 4 | — | |
NHHFHVWZSBAOKB
|
9.0 | IC50 | 3 | — | |
UPRWRNZMVXAVLM
|
9.0 | IC50 | 3 | — | |
WEXJHTQKLRIDBA
|
9.0 | IC50 | 3 | — | |
ZZOVXCVSZXCPAB
|
9.0 | IC50 | 3 | — | |
ZZTQEPNLUZOBOF
|
9.0 | IC50 | 3 | — | |
FLIUGCCDOLARIN
|
9.0 | IC50 | 4 | — | |
HOJKIFJSILSXOV
|
9.0 | IC50 | 3 | — | |
IKPPBUIYPJLCPO
|
9.0 | IC50 | 3 | — | |
LRODNFJRCKXACM
|
9.0 | IC50 | 4 | — | |
RJFSUXPNRYMHRA
|
9.0 | IC50 | 4 | — | |
SGZFQFBJJXRGIS
|
9.0 | IC50 | 4 | — | |
VIXCSOBWOUIQIJ
|
9.0 | IC50 | 3 | — | |
ZZOVXCVSZXCPAB
|
9.0 | IC50 | 3 | — | |
FQGFBVZPDQJURE
|
9.0 | IC50 | 3 | — | |
GUIRLGOCMGPTCZ
|
9.0 | IC50 | 3 | — | |
JMGDTOZRWTXGIB
|
9.0 | IC50 | 4 | — | |
LBJBSCVPRJVYAR
|
9.0 | IC50 | 4 | — | |
LHXGHTSWNSQAAT
|
9.0 | IC50 | 3 | — | |
PXYFMAZFKVHGCP
|
9.0 | IC50 | 4 | — | |
QRZCJVIIIQFGHZ
|
9.0 | IC50 | 3 | — | |
UUKSLYYLPFNFCV
|
9.0 | IC50 | 3 | — | |
VQFVDKZCXCUSNA
|
9.0 | IC50 | 4 | — | |
KTVGSOVNUGSRIM
|
9.0 | IC50 | 3 | — | |
DVBUKYLREULPNY
|
9.0 | IC50 | 3 | — | |
HVZNGQAYECGPHO
|
9.0 | IC50 | 4 | — | |
PQOCNUYHZWCRFU
|
9.0 | IC50 | 4 | — | |
VTMZAPBREHOBOO
|
9.0 | IC50 | 3 | — | |
AAKIPIWTHVPQDP
|
9.0 | IC50 | 3 | — | |
NBQHXIGLUPQFLR
|
9.0 | IC50 | 4 | — | |
YDMCXFWMWSHEBR
|
9.0 | IC50 | 3 | — | |
DUWAWPVUNJBRQD
|
8.9 | IC50 | 4 | — | |
KEMBFYIRAFMFMT
|
8.9 | IC50 | 3 | — | |
PQRRTYZMKUUTSQ
|
8.9 | IC50 | 4 | — |