Target Details
| UniProt AC | P52333 |
|---|---|
| Gene Symbol | JAK3 |
| Protein Name | Tyrosine-protein kinase JAK3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF18379 (FERM_F1) PF18377 (FERM_F2) PF17887 (Jak1_Phl) PF07714 (PK_Tyr_Ser-Thr) PF21990 (SH2_1) |
Summary
- Multi-target molecules 5,161
- Clinical molecules 45
- Avg pChEMBL 7.57
KEGG Pathways (15)
- Chemokine signaling pathway
- Epstein-Barr virus infection
- Hepatitis B
- Human T-cell leukemia virus 1 infection
- JAK-STAT signaling pathway
- Measles
- Necroptosis
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pathways in cancer
- Primary immunodeficiency
- Signaling pathways regulating pluripotency of stem cells
- Th1 and Th2 cell differentiation
- Th17 cell differentiation
- Viral carcinogenesis
Associated Diseases (1)
Active Molecules (5,161)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JYQWFGXKWAXOIK
|
9.3 | IC50 | 3 | — | |
SRVALWZHFUBHNP
|
9.3 | IC50 | 3 | — | |
ACDBOGFFDWLNCX
|
9.3 | IC50 | 2 | — | |
BIUZUMXNKSQCFI
|
9.3 | Ki | 4 | — | |
BTSUQXYEFQQBIJ
|
9.3 | IC50 | 2 | — | |
BWPPEAVIJRXKIH
|
9.3 | IC50 | 2 | — | |
DHJQQONFERYDPZ
|
9.3 | IC50 | 3 | — | |
FSGDGKSWPWYXJK
|
9.3 | IC50 | 2 | — | |
GEGAVKHDOZWMBJ
|
9.3 | IC50 | 2 | — | |
HCMVIWOOWCOZRC
|
9.3 | IC50 | 4 | — | |
HKSZLNNOFSGOKW
|
9.3 | IC50 | 408 | — | |
HVOHXBGDKYDBQD
|
9.3 | IC50 | 2 | — | |
HVOHXBGDKYDBQD
|
9.3 | IC50 | 2 | — | |
IACRSHDPMMMKDK
|
9.3 | IC50 | 3 | — | |
IOJAVMLZYQERBQ
|
9.3 | IC50 | 2 | — | |
KBENESZRTLSKOD
|
9.3 | IC50 | 2 | — | |
KYRQUVYGCZFTQL
|
9.3 | IC50 | 2 | — | |
LJBNEBVTWOQSHN
|
9.3 | IC50 | 2 | — | |
MJHBBCZEVXDESQ
|
9.3 | IC50 | 2 | — | |
MNOGNVQKYDUVPT
|
9.3 | IC50 | 2 | — | |
MOIWQCXOFGXYFZ
|
9.3 | IC50 | 2 | — | |
PCPIKCFUSRCHFD
|
9.3 | IC50 | 2 | — | |
PPRAAYSRROVMEX
|
9.3 | IC50 | 2 | — | |
QCGBDTSLOLLHEJ
|
9.3 | Ki | 4 | — | |
QCGBDTSLOLLHEJ
|
9.3 | Ki | 4 | — | |
QWFFOELVGDLHSA
|
9.3 | IC50 | 2 | — | |
RGEDADHWCUYEEQ
|
9.3 | IC50 | 2 | — | |
UFOROJMBICCFEP
|
9.3 | IC50 | 2 | — | |
UJRAUOKOPQCLEM
|
9.3 | IC50 | 2 | — | |
UUVIRLNTJFTJSY
|
9.3 | IC50 | 2 | — | |
XUZGLJHOFPPBEF
|
9.3 | IC50 | 5 | — | |
XYLKQUBBQYONMI
|
9.3 | IC50 | 2 | — | |
YPCIHFNGHFKCPP
|
9.3 | IC50 | 2 | — | |
YZKHTERFMCPLDP
|
9.3 | IC50 | 2 | — | |
ZRDGJDGEEJEDPT
|
9.3 | IC50 | 2 | — | |
QAUMXKOQGZMGHJ
|
9.3 | IC50 | 3 | — | |
FKKDZJVASSEXKZ
|
9.3 | IC50 | 2 | — | |
KSSGVVODOQPERU
|
9.3 | IC50 | 2 | — | |
MSISQTLXMVHCPT
|
9.3 | IC50 | 4 | — | |
ZROSJPSOILHJQV
|
9.3 | IC50 | 2 | — | |
AARMFTKYYKWETR
|
9.3 | Ki | 4 | — | |
ABHCRSDHBNSQKV
|
9.3 | Ki | 3 | — | |
AECKGAJJKMKUMA
|
9.3 | Ki | 3 | — | |
AIWAMXKDRXZMII
|
9.3 | IC50 | 3 | — | |
AIWSQYMZMZEESE
|
9.3 | Ki | 4 | — | |
AKQUFSFHBPULCX
|
9.3 | Ki | 3 | — | |
AOGXHIHTHRCTPK
|
9.3 | Ki | 2 | — | |
ATKQNWIMTWIHAX
|
9.3 | IC50 | 2 | — | |
ATYDVSUAWJNMMM
|
9.3 | Ki | 3 | — | |
AUIPDNKLZNBXGV
|
9.3 | Ki | 3 | — |