Target Details
| UniProt AC | P52333 |
|---|---|
| Gene Symbol | JAK3 |
| Protein Name | Tyrosine-protein kinase JAK3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF18379 (FERM_F1) PF18377 (FERM_F2) PF17887 (Jak1_Phl) PF07714 (PK_Tyr_Ser-Thr) PF21990 (SH2_1) |
Summary
- Multi-target molecules 5,161
- Clinical molecules 45
- Avg pChEMBL 7.57
KEGG Pathways (15)
- Chemokine signaling pathway
- Epstein-Barr virus infection
- Hepatitis B
- Human T-cell leukemia virus 1 infection
- JAK-STAT signaling pathway
- Measles
- Necroptosis
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pathways in cancer
- Primary immunodeficiency
- Signaling pathways regulating pluripotency of stem cells
- Th1 and Th2 cell differentiation
- Th17 cell differentiation
- Viral carcinogenesis
Associated Diseases (1)
Active Molecules (5,161)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PJTVQALTARBQFE
|
9.5 | Ki | 4 | — | |
VXPVQEJLWUQWPA
|
9.5 | IC50 | 3 | — | |
WIICDYUXOKRMJM
|
9.5 | Ki | 2 | — | |
WIICDYUXOKRMJM
|
9.5 | Ki | 4 | — | |
VZUJWCBHLRHZGN
|
9.5 | IC50 | 2 | — | |
AOOQVVONCAGHIL
|
9.5 | IC50 | 3 | — | |
JUKLRDIBIPCUTH
|
9.5 | IC50 | 2 | — | |
IKURBZUUPLCTRI
|
9.4 | IC50 | 4 | — | |
QMIQJOUVTUIKMM
|
9.4 | IC50 | 3 | — | |
AEDGJZHEZKVHKW
|
9.4 | IC50 | 2 | — | |
JOAGWLAITGLBRM
|
9.4 | IC50 | 3 | — | |
KMHHGCXCFPDSLQ
|
9.4 | IC50 | 2 | — | |
MINAXHKBUIPUJE
|
9.4 | IC50 | 3 | — | |
VVAGTJJOXKEOOR
|
9.4 | IC50 | 2 | — | |
YNOOYZQWHVMQKA
|
9.4 | IC50 | 3 | — | |
ACBQUTNDXICEGK
|
9.4 | IC50 | 2 | — | |
BUAHNPQMVQZWMQ
|
9.4 | IC50 | 2 | — | |
BWVUHOFBASJRGL
|
9.4 | IC50 | 2 | — | |
CATGYHXLDRQPGZ
|
9.4 | IC50 | 3 | — | |
CQVLTKQROAIZOC
|
9.4 | Ki | 4 | — | |
DYNWNZXMEXKEQG
|
9.4 | IC50 | 2 | — | |
FXDHXSDKRXMBJF
|
9.4 | IC50 | 4 | — | |
FYIVGGGCUXWCBN
|
9.4 | IC50 | 2 | — | |
HGMJKEXXCJFENY
|
9.4 | IC50 | 2 | — | |
MHXHZQDDIVMOLK
|
9.4 | IC50 | 2 | — | |
MIEJSPISAIBISA
|
9.4 | IC50 | 2 | — | |
MLABEZYXQDQKQV
|
9.4 | IC50 | 3 | — | |
NDWBUHNJHOUAIV
|
9.4 | IC50 | 2 | — | |
NPXRGBHWBLKOFJ
|
9.4 | Ki | 4 | — | |
OWNKWOSRGVLIAO
|
9.4 | IC50 | 4 | — | |
QBOIBBBYWJLYNM
|
9.4 | IC50 | 2 | — | |
QCSRCAUURQRFKY
|
9.4 | IC50 | 2 | — | |
QGONWVMYZIRRSF
|
9.4 | IC50 | 2 | — | |
QJORGGWPAWDNRO
|
9.4 | IC50 | 2 | — | |
VHTSWIULJUKNRL
|
9.4 | IC50 | 2 | — | |
VMUVVVFKYFIGGE
|
9.4 | IC50 | 2 | — | |
WNIUGDUMLMYFBP
|
9.4 | IC50 | 2 | — | |
ZPDHVAANRIDDBS
|
9.4 | IC50 | 2 | — | |
ZYGSAIOEZWHNPW
|
9.4 | IC50 | 2 | — | |
LLYVJCSGRPQOGO
|
9.4 | IC50 | 4 | — | |
RVUUYYGYSXNUNC
|
9.4 | IC50 | 3 | — | |
OXYLNPXFNFUHGE
|
9.4 | IC50 | 4 | — | |
VRCJTAJIHBPIPH
|
9.4 | IC50 | 3 | — | |
FWXWVZRNYLBRCK
|
9.4 | IC50 | 3 | — | |
WRLLXWRAXRGFBQ
|
9.4 | IC50 | 4 | — | |
YKBQLVVJJHUKDV
|
9.4 | IC50 | 2 | — | |
WVHWGUJFRMEFGH
|
9.3 | IC50 | 3 | — | |
GJMZWYLOARVASY
|
9.3 | IC50 | 6 | — | |
OGJWWUCDNHVDOY
|
9.3 | IC50 | 4 | — | |
HKKFYRPSRCCRQR
|
9.3 | IC50 | 3 | — |