Target Details
| UniProt AC | P52333 |
|---|---|
| Gene Symbol | JAK3 |
| Protein Name | Tyrosine-protein kinase JAK3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF18379 (FERM_F1) PF18377 (FERM_F2) PF17887 (Jak1_Phl) PF07714 (PK_Tyr_Ser-Thr) PF21990 (SH2_1) |
Summary
- Multi-target molecules 5,161
- Clinical molecules 45
- Avg pChEMBL 7.57
KEGG Pathways (15)
- Chemokine signaling pathway
- Epstein-Barr virus infection
- Hepatitis B
- Human T-cell leukemia virus 1 infection
- JAK-STAT signaling pathway
- Measles
- Necroptosis
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pathways in cancer
- Primary immunodeficiency
- Signaling pathways regulating pluripotency of stem cells
- Th1 and Th2 cell differentiation
- Th17 cell differentiation
- Viral carcinogenesis
Associated Diseases (1)
Active Molecules (5,161)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KMGCHJSYIPLBSP
|
9.6 | IC50 | 3 | — | |
PJTVQALTARBQFE
|
9.6 | Ki | 2 | — | |
CKWACTZVXJYDPZ
|
9.5 | IC50 | 3 | — | |
YELDZETVZPUXHI
|
9.5 | IC50 | 3 | — | |
ATIOOYWADXBWPH
|
9.5 | IC50 | 2 | — | |
BEJOSQBBGMLEBM
|
9.5 | IC50 | 3 | — | |
DIBTVUWTGUFWBI
|
9.5 | IC50 | 4 | — | |
DJXKPVCJOOTGHU
|
9.5 | IC50 | 2 | — | |
FNYKNWAPYCCIQE
|
9.5 | IC50 | 3 | — | |
FTIQSPABOXACSR
|
9.5 | IC50 | 3 | — | |
HBAFQIAOOXMYKV
|
9.5 | IC50 | 2 | — | |
HJTWMCDGJVEOQY
|
9.5 | IC50 | 2 | — | |
IJKKBQHULDYNJO
|
9.5 | IC50 | 3 | — | |
IVGXSLJBZRBIIK
|
9.5 | IC50 | 2 | — | |
IYHWPGRNZRXDSS
|
9.5 | IC50 | 2 | — | |
JWLPUQHGINAEID
|
9.5 | IC50 | 2 | — | |
JYKFMRUYKJKTCA
|
9.5 | IC50 | 2 | — | |
KVAOLQZONLRAQP
|
9.5 | IC50 | 2 | — | |
KYLAPPDFIDBGGC
|
9.5 | IC50 | 2 | — | |
LMWZRTIJZLQQJP
|
9.5 | IC50 | 3 | — | |
NSBCDCFIXFFGGR
|
9.5 | IC50 | 2 | — | |
NZXXIWSVVINBQB
|
9.5 | IC50 | 2 | — | |
OHNNRNYUHNGDNO
|
9.5 | IC50 | 15 | — | |
OKNOMBZPAHBAOI
|
9.5 | IC50 | 2 | — | |
OQEHEHLSAFSNPV
|
9.5 | IC50 | 2 | — | |
OYXNZCKLNUECKG
|
9.5 | IC50 | 2 | — | |
PZGWIJSAMUTVLT
|
9.5 | IC50 | 2 | — | |
QIKGVNSHIOKLKZ
|
9.5 | IC50 | 2 | — | |
QNWORZWZMJZYJN
|
9.5 | IC50 | 2 | — | |
RETOGHVZWDPJEU
|
9.5 | IC50 | 2 | — | |
SGJIYRCDJHFJIF
|
9.5 | IC50 | 2 | — | |
SIEMFXMJGAMFQR
|
9.5 | IC50 | 4 | — | |
UFYWHLMLYAFVAN
|
9.5 | IC50 | 3 | — | |
UHJVSLVHPVNWQN
|
9.5 | IC50 | 3 | — | |
UPIXXARGUADGPQ
|
9.5 | IC50 | 2 | — | |
VAAJFRAEGOEUSK
|
9.5 | IC50 | 3 | — | |
WJPORRXQYBLMFT
|
9.5 | IC50 | 2 | — | |
WWQMEXIPGWLRIA
|
9.5 | IC50 | 2 | — | |
WXXVDKLLEOTZPM
|
9.5 | IC50 | 2 | — | |
XDKVRNHZTPJCNO
|
9.5 | IC50 | 2 | — | |
YIGVVPMJPXJTDY
|
9.5 | IC50 | 2 | — | |
YMKKYSADUBPRCK
|
9.5 | IC50 | 2 | — | |
ZUZGPIKWEIVHOP
|
9.5 | IC50 | 2 | — | |
DWSLLEQNJMTLSR
|
9.5 | IC50 | 3 | — | |
GNVJDFYURAVLOR
|
9.5 | IC50 | 3 | — | |
KHSOZOOBSQCDRG
|
9.5 | IC50 | 2 | — | |
AMQJRDKUJJLKCK
|
9.5 | Ki | 2 | — | |
GPOGKSDOWYRIMA
|
9.5 | Ki | 2 | — | |
IKLRDULEVRUACA
|
9.5 | IC50 | 3 | — | |
KQTBXYZYIBLKEB
|
9.5 | IC50 | 3 | — |