Target Details
| UniProt AC | P52333 |
|---|---|
| Gene Symbol | JAK3 |
| Protein Name | Tyrosine-protein kinase JAK3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF18379 (FERM_F1) PF18377 (FERM_F2) PF17887 (Jak1_Phl) PF07714 (PK_Tyr_Ser-Thr) PF21990 (SH2_1) |
Summary
- Multi-target molecules 5,161
- Clinical molecules 45
- Avg pChEMBL 7.57
KEGG Pathways (15)
- Chemokine signaling pathway
- Epstein-Barr virus infection
- Hepatitis B
- Human T-cell leukemia virus 1 infection
- JAK-STAT signaling pathway
- Measles
- Necroptosis
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pathways in cancer
- Primary immunodeficiency
- Signaling pathways regulating pluripotency of stem cells
- Th1 and Th2 cell differentiation
- Th17 cell differentiation
- Viral carcinogenesis
Associated Diseases (1)
Active Molecules (5,161)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FQXJVLSEWHALMZ
|
9.8 | Ki | 2 | — | |
FTQBYQRDFCFCFN
|
9.8 | Ki | 4 | — | |
IMMLXIZVTUKHEQ
|
9.8 | Ki | 4 | — | |
JTQYNUWCYZIYRH
|
9.8 | IC50 | 3 | — | |
JXSIEYYMYPREPS
|
9.8 | IC50 | 3 | — | |
KZPCATSDOZHYDA
|
9.8 | Ki | 4 | — | |
LXCJYFUAMDZSGA
|
9.8 | Ki | 4 | — | |
NNBWJHDKGIUVBS
|
9.8 | Ki | 2 | — | |
NNBWJHDKGIUVBS
|
9.8 | Ki | 2 | — | |
ODJLPNCPBKODCN
|
9.8 | Ki | 2 | — | |
ODJLPNCPBKODCN
|
9.8 | Ki | 4 | — | |
QHHRTNNXPWXSMX
|
9.8 | Ki | 4 | — | |
YEMGRNZLFUZGTR
|
9.8 | IC50 | 2 | — | |
YJSFYJMKVAVFQE
|
9.8 | IC50 | 3 | — | |
LGIBDQRYOFBMTC
|
9.8 | Ki | 6 | Yes | |
LKJRXQYMTPLADK
|
9.8 | IC50 | 3 | — | |
RNXSRQLDXUFACI
|
9.8 | IC50 | 3 | — | |
XEMVVCSEZINFNJ
|
9.8 | IC50 | 2 | — | |
AEYKDHHKLLLVCG
|
9.7 | IC50 | 3 | — | |
HZWSEZYZHCGXGP
|
9.7 | IC50 | 3 | — | |
PLYMRBURAGFOGH
|
9.7 | Ki | 2 | — | |
PLYMRBURAGFOGH
|
9.7 | Ki | 2 | — | |
POMTZDLWTMBAPX
|
9.7 | Ki | 2 | — | |
NYBFBMJGYKYPFD
|
9.7 | IC50 | 3 | — | |
XAPXWXQXXGTZAM
|
9.7 | IC50 | 3 | — | |
ADGZEMSWFJNDIG
|
9.7 | IC50 | 2 | — | |
AMBGBDGUUYGEJS
|
9.7 | Ki | 4 | — | |
AMQJRDKUJJLKCK
|
9.7 | Ki | 4 | — | |
BTDPLPHYTGJMRS
|
9.7 | IC50 | 2 | — | |
BYUXOSCZSBDHCP
|
9.7 | IC50 | 3 | — | |
CQSAMRRIWHJVQQ
|
9.7 | IC50 | 2 | — | |
CQVLTKQROAIZOC
|
9.7 | Ki | 2 | — | |
CTNCYOQZDOTTFX
|
9.7 | IC50 | 3 | — | |
FRZCZWJZDMDTOB
|
9.7 | Ki | 2 | — | |
GJFCCGNALMSJGQ
|
9.7 | IC50 | 2 | — | |
GPOGKSDOWYRIMA
|
9.7 | Ki | 4 | — | |
HBAFQIAOOXMYKV
|
9.7 | IC50 | 2 | — | |
HQOFLQVAJPMMBW
|
9.7 | IC50 | 2 | — | |
HVPQCGSFFCKBQH
|
9.7 | IC50 | 2 | — | |
JMGAJIMHWVWABN
|
9.7 | IC50 | 2 | — | |
JWLPUQHGINAEID
|
9.7 | IC50 | 2 | — | |
JXVIBSHMZHZTST
|
9.7 | IC50 | 3 | — | |
KGSIPBDDGJCGDZ
|
9.7 | IC50 | 2 | — | |
KPLWWYUZVZOXNZ
|
9.7 | IC50 | 2 | — | |
KVAOLQZONLRAQP
|
9.7 | IC50 | 2 | — | |
LKYNKWVSJBBRNP
|
9.7 | Ki | 2 | — | |
MAISEFJAAIILEY
|
9.7 | IC50 | 2 | — | |
MIAKWWNJXPFGAN
|
9.7 | IC50 | 2 | — | |
NFABHXGDHDFKDI
|
9.7 | IC50 | 2 | — | |
NPIRZUMAGGQJIG
|
9.7 | IC50 | 2 | — |