Target Details
| UniProt AC | P51957 |
|---|---|
| Gene Symbol | NEK4 |
| Protein Name | Serine/threonine-protein kinase Nek4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 71
- Clinical molecules 3
- Avg pChEMBL 6.6
Active Molecules (71)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KAKFXRYHYUPXSU
|
6.1 | Ki | 16 | — | |
KNACLJBHKVSTDL
|
6.1 | Ki | 40 | — | |
MQRDVGBWWVWMEN
|
6.1 | Ki | 47 | — | |
NWAUBAGBGOPJLF
|
6.1 | Ki | 51 | Yes | |
OUJZYQBEFNDJQN
|
6.1 | Ki | 71 | — | |
OWDRQHVEJIYVOI
|
6.1 | Ki | 47 | — | |
PTVPBWWDGZSEAF
|
6.1 | Ki | 63 | — | |
SBFPHSVZEXSHTL
|
6.1 | Ki | 62 | — | |
SUULIUKTZNKMMB
|
6.1 | Ki | 10 | — | |
SYLTYCLPHHSEIJ
|
6.1 | Ki | 27 | — | |
XSRHBCYNCKAFKS
|
6.1 | Ki | 45 | — | |
DJLORVJVWIBDME
|
6.0 | Ki | 24 | — | |
HEUSUIRCBWROMH
|
6.0 | Ki | 64 | — | |
IMHKMKWSWHFKTM
|
6.0 | IC50 | 13 | — | |
JAMDNXUAYUHJLJ
|
6.0 | Ki | 40 | — | |
JZTOUVBEZONDKA
|
6.0 | Ki | 80 | — | |
KRIUNPBAQZGFQA
|
6.0 | Ki | 76 | — | |
XQVVPGYIWAGRNI
|
6.0 | Ki | 19 | — | |
YDWMUCKJUNLURC
|
6.0 | IC50 | 24 | — | |
YWTBGJGMTBHQTM
|
6.0 | Ki | 65 | — | |
ZGZVRPRSFXRGCF
|
6.0 | Ki | 76 | — |