Target Details
| UniProt AC | P51956 |
|---|---|
| Gene Symbol | NEK3 |
| Protein Name | Serine/threonine-protein kinase Nek3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 8
- Clinical molecules 0
- Avg pChEMBL 6.21
Active Molecules (8)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NHHQJBCNYHBUSI
|
6.8 | Kd | 220 | — | |
ATWJOSDBVRWRHS
|
6.6 | IC50 | 5 | — | |
JOOXLOJCABQBSG
|
6.2 | Kd | 139 | — | |
XQVVPGYIWAGRNI
|
6.1 | Kd | 34 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
YYLKKYCXAOBSRM
|
6.0 | Kd | 191 | — |