Target Details
| UniProt AC | P51955 |
|---|---|
| Gene Symbol | NEK2 |
| Protein Name | Serine/threonine-protein kinase Nek2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 120
- Clinical molecules 13
- Avg pChEMBL 6.6
Associated Diseases (1)
Active Molecules (120)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RYYNGWLOYLRZLK
|
6.1 | Ki | 104 | — | |
YMIJUBCSOKSFRU
|
6.1 | Ki | 87 | — | |
KWJAATQOHSNKKF
|
6.0 | IC50 | 3 | — | |
LYADGAGFYYXXIO
|
6.0 | IC50 | 82 | — | |
CUIHSIWYWATEQL
|
6.0 | Kd | 61 | Yes | |
AQKQATGZIKRZMQ
|
6.0 | Ki | 16 | — | |
BRTHUECZMVKNMQ
|
6.0 | Ki | 31 | — | |
FQYLJBVSYHZWLT
|
6.0 | Ki | 35 | Yes | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
JSDGKSMNPHJDFK
|
6.0 | Ki | 35 | — | |
JVUYFKGAACUDSV
|
6.0 | IC50 | 2 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
NECQZMQPXFYVOY
|
6.0 | Ki | 26 | — | |
NLUPJKQOKWBWFC
|
6.0 | Ki | 69 | — | |
PCQMERRARZKTPW
|
6.0 | Ki | 68 | — | |
QKPLUKMJEKRAJD
|
6.0 | Ki | 30 | Yes | |
SFPWNTQWFFNJIH
|
6.0 | Ki | 48 | — | |
XCHWBXBDZRJVDP
|
6.0 | Ki | 51 | — | |
ZXLFIHLBHMLHFJ
|
6.0 | Ki | 31 | — |