Target Details
| UniProt AC | P51955 |
|---|---|
| Gene Symbol | NEK2 |
| Protein Name | Serine/threonine-protein kinase Nek2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 120
- Clinical molecules 13
- Avg pChEMBL 6.6
Associated Diseases (1)
Active Molecules (120)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZHJGWYRLJUCMRT
|
6.6 | Kd | 18 | — | |
APPXQUDJLJXULP
|
6.6 | IC50 | 47 | — | |
JWNPDZNEKVCWMY
|
6.6 | IC50 | 57 | Yes | |
RDAXOPGNTONHMU
|
6.5 | IC50 | 2 | — | |
XKZQZMSAWVDRSP
|
6.5 | IC50 | 39 | Yes | |
CKVWQORGCCEYHS
|
6.5 | Ki | 50 | — | |
MQRDVGBWWVWMEN
|
6.5 | Ki | 47 | — | |
NFKMFNBKEOQNPZ
|
6.5 | Ki | 43 | — | |
QVNZKVACBBTKSL
|
6.5 | Ki | 38 | — | |
UQNNJYLAPYGZBD
|
6.5 | Ki | 28 | — | |
XOOAAYRIVATZNM
|
6.5 | Ki | 55 | — | |
HKZKELVPGXJIMW
|
6.4 | Ki | 41 | — | |
LGHBDVLAHHANMX
|
6.4 | Ki | 53 | — | |
NRGYZNJPCGRCLV
|
6.4 | Ki | 52 | — | |
NWAUBAGBGOPJLF
|
6.4 | Ki | 51 | Yes | |
ULHGAQSVFPOUDY
|
6.4 | Ki | 43 | — | |
VSVWQTDDGQSGHP
|
6.4 | Ki | 51 | — | |
CKNBSSMNQGLXEA
|
6.3 | Kd | 3 | — | |
JTSLALYXYSRPGW
|
6.3 | Kd | 8 | — | |
AEYLJTAIDDIOBA
|
6.3 | Ki | 53 | — | |
DKSNLQYRZJKYOC
|
6.3 | Ki | 51 | — | |
GSXRCPJTNIGKSZ
|
6.3 | Ki | 43 | — | |
JCFJQIHDZHHMQT
|
6.3 | Ki | 42 | — | |
JSKUWFIZUALZLX
|
6.3 | Ki | 33 | — | |
NFMGZVPRGVERNN
|
6.3 | Ki | 44 | — | |
NKGLJTITEFZKAN
|
6.3 | Ki | 35 | — | |
PIQCTGMSNWUMAF
|
6.3 | Ki | 137 | Yes | |
WINHZLLDWRZWRT
|
6.3 | Kd | 201 | Yes | |
ZGDSBEUMPIMXBM
|
6.3 | Ki | 42 | — | |
OYONTEXKYJZFHA
|
6.2 | Kd | 69 | Yes | |
DZSUJUOJJJCWGG
|
6.2 | Ki | 55 | Yes | |
FPQHXFMYXQZPSV
|
6.2 | Ki | 23 | — | |
GCYXEGSPUDSZJY
|
6.2 | Ki | 82 | — | |
HRZOUBQYVUXBNS
|
6.2 | Ki | 38 | — | |
HSKVRPZJBMXFDX
|
6.2 | Ki | 20 | — | |
JAMDNXUAYUHJLJ
|
6.2 | Ki | 40 | — | |
RJZDECGDCKOHBV
|
6.2 | Ki | 70 | — | |
RKKIDHHGKNGTQI
|
6.2 | Ki | 28 | — | |
RYAVJHIPOWNWDE
|
6.2 | Ki | 38 | — | |
XAYDUCQADQTDGX
|
6.2 | Ki | 12 | — | |
BNJAETMQKIKKSN
|
6.2 | IC50 | 2 | — | |
WVUNYSQLFKLYNI
|
6.2 | Kd | 46 | Yes | |
HKSZLNNOFSGOKW
|
6.1 | Kd | 408 | — | |
HKSZLNNOFSGOKW
|
6.1 | Kd | 213 | — | |
CNTCGRJDUJEUDG
|
6.1 | Ki | 37 | — | |
GXJSLIOOPZRPEV
|
6.1 | Ki | 34 | — | |
JHYHWHUTTXJICB
|
6.1 | Ki | 18 | — | |
KKYPRNBBPBRJQX
|
6.1 | Ki | 40 | — | |
QQWUGDVOUVUTOY
|
6.1 | Ki | 231 | Yes | |
RUPJOKGREQMQSI
|
6.1 | Ki | 9 | — |