Target Details
UniProt ACP51948
Gene SymbolMNAT1
Protein NameCDK-activating kinase assembly factor MAT1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF25811 (CAK-anch_MAT1) PF06391 (MAT1) PF17121 (zf-C3HC4_5)
Summary
  • Multi-target molecules 448
  • Clinical molecules 7
  • Avg pChEMBL 7.1
Top Co-occurrence Targets
Active Molecules (448)
InChIKey pChEMBL Type Targets Clinical
PEMUGDMSUDYLHU 8.9 IC50 5
GWRVGNYOXQHPMF 8.7 Ki 5
KPABJHHKKJIDGX 8.7 Ki 3
ODTNVBQMSINVPK 8.7 Ki 6
GLOFAMHSVMGLKL 8.6 IC50 4
JDJOUBVVSQDIRC 8.6 IC50 3
CSYVEHWJTGNMOY 8.6 Ki 7
XSKBBXDFCDHKGM 8.5 Ki 3
ODTNVBQMSINVPK 8.5 Ki 6
YCVGLKWJKIKVBI 8.5 Ki 6
CWZJJLMGMPZMDY 8.4 IC50 3
VZQDFIKUYBSQRQ 8.3 IC50 6
ZBFCXGKZXRBIFF 8.3 IC50 5
UZPUYHARAXYZLT 8.2 IC50 3
XAQRVVLOLCCQEB 8.2 IC50 3
DHZKWPMYADCRCR 8.2 IC50 4
QMNWYIJJYDNVOQ 8.2 IC50 3
VWSDWOYFAZHKHK 8.2 IC50 3
WINYZTMONKJGNR 8.2 IC50 3
IVOIFGRBXZVOFK 8.2 IC50 3
AYCPARAPKDAOEN 8.2 IC50 73
KOBLEPSVVLTMLE 8.1 IC50 3
LHGBWMYXJKRMIP 8.1 IC50 3
FPTHHKVHJDUFEA 8.1 IC50 3
IOKORVXLSWJWQL 8.1 IC50 3
VBYGXNURPHQSPG 8.1 IC50 5
JWLWJKKNZAGESY 8.1 IC50 3
VBNZZGDQJYVFDA 8.1 IC50 3
CGPMSCGCDRRRHS 8.1 IC50 3
ZCCPLJOKGAACRT 8.1 Kd 599
JOPQDQBLBCRZES 8.1 IC50 3
QESKJLNPFAAHST 8.1 IC50 3
ROBBURZERULYQU 8.1 IC50 3
OIXCMADAZITJOX 8.1 IC50 3
JVBMCKNTDXXCTA 8.0 IC50 3
MZVXBMQKLXUJEV 8.0 IC50 3
FGNHJXSBQQICEW 8.0 Ki 7
KPABJHHKKJIDGX 8.0 IC50 3
ZMFBLJJBZOWLHV 8.0 IC50 3
LGHAAIHVITWSPZ 8.0 IC50 3
VXBAJLGYBMTJCY 8.0 IC50 34 Yes
KMCFZYFLOLCIFG 8.0 IC50 3
OZIBOKYMPVXMRJ 8.0 IC50 3
GLMORIZVXAPSPO 8.0 IC50 3
SOHKYLNCPBLXTM 7.9 IC50 3
DQDNKGFWJQBIFN 7.9 IC50 3
UOMFAOIPQSGEDO 7.9 IC50 3
OVBAZPDZTDYHBW 7.9 IC50 3
FONRCZUZCHXWBD 7.9 IC50 8
KPLAOBBKVKBAHH 7.9 IC50 3
2D structure