Target Details
| UniProt AC | P51948 |
|---|---|
| Gene Symbol | MNAT1 |
| Protein Name | CDK-activating kinase assembly factor MAT1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF25811 (CAK-anch_MAT1) PF06391 (MAT1) PF17121 (zf-C3HC4_5) |
Summary
- Multi-target molecules 448
- Clinical molecules 7
- Avg pChEMBL 7.1
KEGG Pathways (2)
Active Molecules (448)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PEMUGDMSUDYLHU
|
8.9 | IC50 | 5 | — | |
GWRVGNYOXQHPMF
|
8.7 | Ki | 5 | — | |
KPABJHHKKJIDGX
|
8.7 | Ki | 3 | — | |
ODTNVBQMSINVPK
|
8.7 | Ki | 6 | — | |
GLOFAMHSVMGLKL
|
8.6 | IC50 | 4 | — | |
JDJOUBVVSQDIRC
|
8.6 | IC50 | 3 | — | |
CSYVEHWJTGNMOY
|
8.6 | Ki | 7 | — | |
XSKBBXDFCDHKGM
|
8.5 | Ki | 3 | — | |
ODTNVBQMSINVPK
|
8.5 | Ki | 6 | — | |
YCVGLKWJKIKVBI
|
8.5 | Ki | 6 | — | |
CWZJJLMGMPZMDY
|
8.4 | IC50 | 3 | — | |
VZQDFIKUYBSQRQ
|
8.3 | IC50 | 6 | — | |
ZBFCXGKZXRBIFF
|
8.3 | IC50 | 5 | — | |
UZPUYHARAXYZLT
|
8.2 | IC50 | 3 | — | |
XAQRVVLOLCCQEB
|
8.2 | IC50 | 3 | — | |
DHZKWPMYADCRCR
|
8.2 | IC50 | 4 | — | |
QMNWYIJJYDNVOQ
|
8.2 | IC50 | 3 | — | |
VWSDWOYFAZHKHK
|
8.2 | IC50 | 3 | — | |
WINYZTMONKJGNR
|
8.2 | IC50 | 3 | — | |
IVOIFGRBXZVOFK
|
8.2 | IC50 | 3 | — | |
AYCPARAPKDAOEN
|
8.2 | IC50 | 73 | — | |
KOBLEPSVVLTMLE
|
8.1 | IC50 | 3 | — | |
LHGBWMYXJKRMIP
|
8.1 | IC50 | 3 | — | |
FPTHHKVHJDUFEA
|
8.1 | IC50 | 3 | — | |
IOKORVXLSWJWQL
|
8.1 | IC50 | 3 | — | |
VBYGXNURPHQSPG
|
8.1 | IC50 | 5 | — | |
JWLWJKKNZAGESY
|
8.1 | IC50 | 3 | — | |
VBNZZGDQJYVFDA
|
8.1 | IC50 | 3 | — | |
CGPMSCGCDRRRHS
|
8.1 | IC50 | 3 | — | |
ZCCPLJOKGAACRT
|
8.1 | Kd | 599 | — | |
JOPQDQBLBCRZES
|
8.1 | IC50 | 3 | — | |
QESKJLNPFAAHST
|
8.1 | IC50 | 3 | — | |
ROBBURZERULYQU
|
8.1 | IC50 | 3 | — | |
OIXCMADAZITJOX
|
8.1 | IC50 | 3 | — | |
JVBMCKNTDXXCTA
|
8.0 | IC50 | 3 | — | |
MZVXBMQKLXUJEV
|
8.0 | IC50 | 3 | — | |
FGNHJXSBQQICEW
|
8.0 | Ki | 7 | — | |
KPABJHHKKJIDGX
|
8.0 | IC50 | 3 | — | |
ZMFBLJJBZOWLHV
|
8.0 | IC50 | 3 | — | |
LGHAAIHVITWSPZ
|
8.0 | IC50 | 3 | — | |
VXBAJLGYBMTJCY
|
8.0 | IC50 | 34 | Yes | |
KMCFZYFLOLCIFG
|
8.0 | IC50 | 3 | — | |
OZIBOKYMPVXMRJ
|
8.0 | IC50 | 3 | — | |
GLMORIZVXAPSPO
|
8.0 | IC50 | 3 | — | |
SOHKYLNCPBLXTM
|
7.9 | IC50 | 3 | — | |
DQDNKGFWJQBIFN
|
7.9 | IC50 | 3 | — | |
UOMFAOIPQSGEDO
|
7.9 | IC50 | 3 | — | |
OVBAZPDZTDYHBW
|
7.9 | IC50 | 3 | — | |
FONRCZUZCHXWBD
|
7.9 | IC50 | 8 | — | |
KPLAOBBKVKBAHH
|
7.9 | IC50 | 3 | — |