Target Details
| UniProt AC | P51946 |
|---|---|
| Gene Symbol | CCNH |
| Protein Name | Cyclin-H |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF16899 (Cyclin_C_2) PF00134 (Cyclin_N) |
Summary
- Multi-target molecules 744
- Clinical molecules 17
- Avg pChEMBL 7.03
KEGG Pathways (3)
Active Molecules (744)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KAUXKMRRDIDIRK
|
10.5 | Kd | 8 | — | |
DQFXKZPDQHUJLY
|
10.2 | Kd | 8 | — | |
JDJOUBVVSQDIRC
|
10.2 | Kd | 3 | — | |
NUMHIIKAGFNIFT
|
10.2 | Kd | 8 | — | |
DGAWYBIEBJUVHR
|
10.1 | Kd | 8 | — | |
DIIRGFRZMVBYSW
|
10.1 | Kd | 8 | — | |
PCHKTFSWKCJOTQ
|
10.1 | Kd | 8 | — | |
JEWRIBSMLSEECE
|
10.0 | Kd | 8 | — | |
XNWQJSPBCYZFAU
|
10.0 | Kd | 8 | — | |
QVBVFLKFEISMLZ
|
9.8 | Kd | 9 | — | |
SLIFZZITPODXKX
|
9.8 | Kd | 6 | — | |
BFEWHEFVBQRIIR
|
9.7 | Kd | 8 | — | |
XWKQZYOSWGEGIH
|
9.5 | Kd | 9 | — | |
YDHKLKQGRRFWHD
|
9.5 | Kd | 8 | — | |
HZZNUWNFLHMBRW
|
9.4 | Kd | 9 | — | |
CVWXJKQAOSCOAB
|
9.2 | IC50 | 35 | — | |
MAUGWAUUEVZZEV
|
9.0 | IC50 | 3 | — | |
TWWKXZDIDHDHRF
|
9.0 | IC50 | 7 | — | |
YISMQBFJYDFMAL
|
9.0 | IC50 | 46 | — | |
GQSVAEJGZAOKMN
|
8.9 | IC50 | 2 | — | |
PEMUGDMSUDYLHU
|
8.9 | IC50 | 5 | — | |
RVZJFCNYSSUDCU
|
8.9 | IC50 | 7 | — | |
XLSYZSRXVVCHLS
|
8.7 | IC50 | 48 | — | |
GWRVGNYOXQHPMF
|
8.7 | Ki | 5 | — | |
KPABJHHKKJIDGX
|
8.7 | Ki | 3 | — | |
ODTNVBQMSINVPK
|
8.7 | Ki | 6 | — | |
PSXIVNJKJRIQFT
|
8.7 | IC50 | 2 | — | |
GLOFAMHSVMGLKL
|
8.6 | IC50 | 4 | — | |
WDLJRFFGBASGDH
|
8.6 | IC50 | 2 | — | |
CSYVEHWJTGNMOY
|
8.6 | Ki | 7 | — | |
XSKBBXDFCDHKGM
|
8.5 | Ki | 3 | — | |
ODTNVBQMSINVPK
|
8.5 | Ki | 6 | — | |
YCVGLKWJKIKVBI
|
8.5 | Ki | 6 | — | |
CWZJJLMGMPZMDY
|
8.4 | IC50 | 3 | — | |
AUIDPIHWVJVXJZ
|
8.3 | IC50 | 4 | — | |
VZQDFIKUYBSQRQ
|
8.3 | IC50 | 6 | — | |
ZBFCXGKZXRBIFF
|
8.3 | IC50 | 5 | — | |
UZPUYHARAXYZLT
|
8.2 | IC50 | 3 | — | |
YBLOCRXWYOGVKP
|
8.2 | IC50 | 2 | — | |
UUMGQHGVBRZLJI
|
8.2 | IC50 | 2 | — | |
XAQRVVLOLCCQEB
|
8.2 | IC50 | 3 | — | |
IJIGRXABGQBDBA
|
8.2 | Ki | 10 | — | |
DHZKWPMYADCRCR
|
8.2 | IC50 | 4 | — | |
PFRRCIUUGVFNKY
|
8.2 | IC50 | 3 | — | |
QMNWYIJJYDNVOQ
|
8.2 | IC50 | 3 | — | |
UFZVUCDJZZJPMF
|
8.2 | IC50 | 3 | — | |
VWSDWOYFAZHKHK
|
8.2 | IC50 | 3 | — | |
WINYZTMONKJGNR
|
8.2 | IC50 | 3 | — | |
IVOIFGRBXZVOFK
|
8.2 | IC50 | 3 | — | |
AYCPARAPKDAOEN
|
8.2 | IC50 | 73 | — |