Target Details
UniProt ACP51817
Gene SymbolPRKX
Protein NamecAMP-dependent protein kinase catalytic subunit PRKX
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00069 (Pkinase)
Summary
  • Multi-target molecules 209
  • Clinical molecules 6
  • Avg pChEMBL 7.02
Top Co-occurrence Targets
Active Molecules (209)
InChIKey pChEMBL Type Targets Clinical
NGDNKYRUKIPCLK 6.4 Ki 12
NOBMKUVHFRVBES 6.4 Ki 19
OUJZYQBEFNDJQN 6.4 Ki 71
OWDRQHVEJIYVOI 6.4 Ki 47
PMXKUMCLYSFPJB 6.4 IC50 4
UIRCQOKSJDLYBB 6.4 Ki 50
UQNNJYLAPYGZBD 6.4 Ki 28
VSVWQTDDGQSGHP 6.4 Ki 51
ZPVLRSVLOWVDJC 6.4 Ki 14
DWTNLZZEPSCAIH 6.3 Ki 25
JBLPUDJLELBRHC 6.3 Ki 9
LNYJUWCJKQGEPR 6.3 Ki 3
MASJMHFQMYAPJR 6.3 Ki 41
MDJCUXFFMNEBHG 6.3 Ki 13
OMKZJNFKGWJFNX 6.3 Ki 8
PCQMERRARZKTPW 6.3 Ki 68
QFHRPRDSAHFZEG 6.3 Ki 6
XZZUBMJMGJRIKY 6.3 Ki 4
DGLFSNZWRYADFC 6.2 IC50 12
DJUSDFVEBBYFFL 6.2 Ki 27
KXPTUMLQPMMHGT 6.2 IC50 4
AEYLJTAIDDIOBA 6.2 Ki 53
DKXHSOUZPMHNIZ 6.2 Ki 51 Yes
IYOZTVGMEWJPKR 6.2 Ki 10
JJTYLBBKGQOISV 6.2 Ki 15
KAKGFGCTONHQJW 6.2 Ki 25
KXPWWMPXNUOYOH 6.2 Ki 24
RIBBPSYZBQQTQC 6.2 Ki 15
ZGDYBJXDIXVTLV 6.2 Ki 54
BUDOGSSTKVVWDR 6.1 Ki 8
CRKQBJZCCHKEGI 6.1 Ki 20
DCTBPIBEQFLAOQ 6.1 Ki 13
FBWWNLBZZFVRQY 6.1 Ki 4
KVYKDXMRLMPSGQ 6.1 Ki 7
LCGSWTFWYNYUKS 6.1 Ki 26
LRLDYTTWQIFWBD 6.1 Ki 25
MZDKLVOWGIOKTN 6.1 Ki 80
NFMGZVPRGVERNN 6.1 Ki 44
NRSGWEVTVGZDFC 6.1 Ki 50
PFCUZXCHLYIMTJ 6.1 Ki 18
PYXQMJSGJIJHJT 6.1 Ki 28
STUPRWVTVIXNLF 6.1 Ki 6
TWCARTFPHQNBPF 6.1 Ki 16
UTQPKPHUIMHAAN 6.1 Ki 22
BMGQWWVMWDBQGC 6.0 Kd 147 Yes
AQKQATGZIKRZMQ 6.0 Ki 16
IVVSBEQDCAZLFY 6.0 IC50 333
JMIIFJIJWDCOEP 6.0 Ki 15
JSKUWFIZUALZLX 6.0 Ki 33
KHVVJKLNKLQLJZ 6.0 IC50 288
2D structure