Target Details
| UniProt AC | P51817 |
|---|---|
| Gene Symbol | PRKX |
| Protein Name | cAMP-dependent protein kinase catalytic subunit PRKX |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 209
- Clinical molecules 6
- Avg pChEMBL 7.02
Active Molecules (209)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MSROHJGQUMVBTJ
|
7.5 | IC50 | 3 | — | |
ACSYKUPGCXYRRO
|
7.5 | Ki | 26 | — | |
BGYVWFZMYBWCNY
|
7.5 | Ki | 30 | — | |
NCQQZIOVNVXPQY
|
7.5 | IC50 | 4 | — | |
OHPRWVPOPFGLJG
|
7.5 | Ki | 19 | — | |
SLKCVFPEQGHNSI
|
7.5 | Ki | 29 | — | |
XPHWIERLJBFPFV
|
7.5 | Ki | 69 | — | |
GLXJGZLTPLOTJM
|
7.5 | IC50 | 4 | — | |
FYRQDEVTRMEZHR
|
7.4 | Ki | 7 | — | |
IJNGXROUMFEKDB
|
7.4 | Ki | 39 | — | |
JRVSFZKYQCETAH
|
7.4 | Ki | 19 | — | |
NWMPVMMGSHXANZ
|
7.4 | Ki | 58 | — | |
VVEGARMQKNYDID
|
7.4 | Ki | 24 | — | |
XSRHBCYNCKAFKS
|
7.4 | Ki | 45 | — | |
YPJJSXBVVGPFHA
|
7.4 | Ki | 18 | — | |
ZGGIYFOLDBTZIL
|
7.4 | Ki | 27 | — | |
ZKLJKKASNXVQBZ
|
7.4 | Ki | 27 | — | |
UIARLYUEJFELEN
|
7.4 | Kd | 289 | Yes | |
NXSJMRCTGYTSTK
|
7.4 | Kd | 200 | — | |
FDBPGAHVEGEARY
|
7.3 | Ki | 19 | — | |
HSMUWLLZAZCLHF
|
7.3 | Ki | 25 | — | |
KCKXYZOBGBJZEG
|
7.3 | Ki | 36 | — | |
NGOGFTYYXHNFQH
|
7.3 | Ki | 15 | — | |
QVWKRMXAYICTFS
|
7.3 | Ki | 8 | — | |
XSDJOIOVIMPMHD
|
7.3 | Ki | 44 | — | |
YOVNFNXUCOWYSG
|
7.3 | Ki | 33 | Yes | |
ZGZVRPRSFXRGCF
|
7.3 | Ki | 76 | — | |
ZRQXCQXWTLVASO
|
7.3 | Ki | 36 | — | |
ZYTFPHRVOZXPGZ
|
7.3 | Ki | 30 | — | |
UBZNLGBMKJHEFB
|
7.2 | IC50 | 3 | — | |
FUMCKNCUEAQHCV
|
7.2 | Ki | 103 | — | |
LPILBMJJRGTKOQ
|
7.2 | Ki | 27 | — | |
SHENEEFOURUIBP
|
7.2 | Ki | 29 | — | |
YWTBGJGMTBHQTM
|
7.2 | Ki | 65 | — | |
ZCXXFPLQFFRMPN
|
7.2 | Ki | 12 | — | |
KEWARFUPGHEOFW
|
7.1 | IC50 | 3 | — | |
LACOMQAWPSFXQC
|
7.1 | Ki | 27 | — | |
SNQKPKFVSANKFP
|
7.1 | IC50 | 6 | — | |
UDFDIIVNIYWXDM
|
7.1 | Ki | 74 | — | |
XFWUTMHVDGPWLH
|
7.1 | Ki | 75 | — | |
BPNUQXPIQBZCMR
|
7.0 | Kd | 83 | Yes | |
CYLGCMABIBXHIQ
|
7.0 | Ki | 16 | — | |
GQLWKGVBOIYMTN
|
7.0 | Ki | 35 | — | |
KCLZJAVIQDVQCK
|
7.0 | Ki | 5 | — | |
KNVOICXEDILAGT
|
7.0 | Ki | 17 | — | |
OWRXHGAFWZFFCW
|
7.0 | Ki | 113 | — | |
SKKRZILJUKYLJS
|
7.0 | Ki | 25 | — | |
URNZTLZSAVLTIZ
|
7.0 | Ki | 26 | — | |
WVFWTUJEHMVUBG
|
7.0 | Ki | 25 | — | |
GJOXRIYWDHESDF
|
6.9 | Ki | 27 | — |