Target Details
UniProt ACP51817
Gene SymbolPRKX
Protein NamecAMP-dependent protein kinase catalytic subunit PRKX
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00069 (Pkinase)
Summary
  • Multi-target molecules 209
  • Clinical molecules 6
  • Avg pChEMBL 7.02
Top Co-occurrence Targets
Active Molecules (209)
InChIKey pChEMBL Type Targets Clinical
HKSZLNNOFSGOKW 9.5 Ki 118
NJPWCTYVEJIQBM 9.0 Ki 72
XYZNKCSDQRKAFR 9.0 Ki 53
HNXJWWRRSGDVIW 8.9 Ki 13
NPLQZQGAZAUUTB 8.9 Ki 9
HKSZLNNOFSGOKW 8.8 IC50 408
BEJCLDKQCNVTQR 8.8 Ki 16
MTYMWGNJKDHWGN 8.8 Ki 18
ZKHDDJKHTPLPOQ 8.8 Ki 62
HOYRWTWZUFFACV 8.7 Ki 28
SRONQUHCRFZABC 8.6 Ki 28
YGEACCLUBSGMMJ 8.6 Ki 16
LRZYYIZFBXFSJB 8.5 Ki 69
WDARYLSSWBWVCU 8.5 Ki 49
XNWKXXIGSPPPBH 8.5 Ki 31
DQPYZHUAILXFJI 8.4 Ki 27
NEWAULHLLUCDPD 8.4 Ki 27
AOBLBPWPSKBHSI 8.3 Ki 55
PLHUMPJXRHMFFR 8.3 Ki 28
VXYDJXMHISGSDA 8.3 Ki 59
ADMFLILDQJSEIK 8.2 Ki 72
LHQWPYOYDRVMFI 8.2 Ki 21
QATMNAAQTUISJK 8.2 Ki 13
QTMFCQXLQBJZQU 8.2 IC50 4
KGPGFQWBCSZGEL 8.1 Kd 59 Yes
ZDTUVVAJVVQVOT 8.1 IC50 4
BSFNGHCTZDCQBF 8.1 Ki 93
SYSUZXPGQXEWCZ 8.1 Ki 10
MIYRKQLKDQNUKZ 8.0 Ki 23
RGOPHVZLEMGMBZ 8.0 Ki 20
XXSPHNFKLDJDAK 8.0 Ki 26
RWKDVIAVTRRJIR 7.9 Ki 23
UPPGGRZNGRFDAU 7.9 Ki 21
XZONYYFHQICDAM 7.9 Ki 19
AWDORCFLUJZUQS 7.8 Ki 22
BPNUQXPIQBZCMR 7.7 Ki 60
KHGPYYFCIAISBU 7.7 Ki 31
LSLPDHNUWRDOGC 7.7 Ki 25
LXVBELDBJGYFEM 7.7 Ki 20
PHWHNHYZZNJPLB 7.7 Ki 16
SMRWVXLSRJWVBF 7.7 Ki 25
UYGYYOIUVFMGKQ 7.7 Ki 30
XFTPNRUQKBIHDT 7.7 Ki 8
KTWBYGUSEYSRND 7.6 Ki 28
PUYIXDDMOUMMRR 7.6 Ki 27
RFBPWKMQWSIPEO 7.6 Ki 28
SGHXFHRRWFLILP 7.6 Ki 29
XMFUGSRATNLPRM 7.6 Ki 19
XUFLBSMTYMFOQH 7.6 Ki 43
JJTVMBJRPZIZDA 7.6 IC50 4
2D structure