Target Details
| UniProt AC | P51813 |
|---|---|
| Gene Symbol | BMX |
| Protein Name | Cytoplasmic tyrosine-protein kinase BMX |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00779 (BTK) PF00169 (PH) PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) |
Summary
- Multi-target molecules 226
- Clinical molecules 11
- Avg pChEMBL 7.47
Active Molecules (226)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RDTDWGQDFJPTPD
|
6.4 | IC50 | 6 | Yes | |
DNXDQVLTWZNPEQ
|
6.4 | IC50 | 3 | — | |
QNABDSWBQJKBHK
|
6.4 | IC50 | 45 | — | |
VJDVKRQPRSCAPE
|
6.3 | IC50 | 2 | — | |
ABSANYKJICYHQP
|
6.3 | IC50 | 4 | — | |
CUABMPOJOBCXJI
|
6.3 | Kd | 3 | — | |
CBRJPFGIXUFMTM
|
6.2 | IC50 | 7 | — | |
LSEAQLOYCHTEOK
|
6.2 | IC50 | 10 | — | |
VSFINVOSLLRTIP
|
6.2 | IC50 | 6 | — | |
ZFKQQXLECNVLOF
|
6.2 | IC50 | 7 | — | |
MFAQYJIYDMLAIM
|
6.2 | Kd | 130 | Yes | |
NXSJMRCTGYTSTK
|
6.2 | Kd | 200 | — | |
WDTHDWKPTWWHLS
|
6.2 | IC50 | 13 | — | |
UORAPQCBWYIISR
|
6.1 | Kd | 2 | — | |
YQYNAUOOJUVDPB
|
6.1 | Kd | 3 | — | |
GUBJNPWVIUFSTR
|
6.1 | Kd | 103 | — | |
HGYLDYXQKAISMX
|
6.1 | Kd | 4 | — | |
LGIHMFDYIKUOSS
|
6.1 | IC50 | 2 | — | |
CJQGLUJHMXCLQY
|
6.1 | IC50 | 11 | — | |
OSVUGUHRKMMBSE
|
6.1 | Kd | 170 | — | |
WIZIQUFUGUEWKY
|
6.1 | IC50 | 6 | — | |
AUUIJHXHLCNNBO
|
6.1 | IC50 | 3 | — | |
KDYQGXDLDYYRDX
|
6.0 | IC50 | 2 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |