Target Details
| UniProt AC | P51813 |
|---|---|
| Gene Symbol | BMX |
| Protein Name | Cytoplasmic tyrosine-protein kinase BMX |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00779 (BTK) PF00169 (PH) PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) |
Summary
- Multi-target molecules 226
- Clinical molecules 11
- Avg pChEMBL 7.47
Active Molecules (226)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZJSNZHATZAWKIQ
|
7.0 | Kd | 5 | — | |
BAYUMEAMGPZXKA
|
7.0 | IC50 | 3 | — | |
AHGUJKCTSXOYES
|
7.0 | IC50 | 4 | — | |
ZZQMSKHNPZIQCU
|
7.0 | IC50 | 3 | — | |
YPXWUKLQAUBCPF
|
7.0 | IC50 | 8 | — | |
RVCKMZIQUFKZFD
|
7.0 | IC50 | 7 | — | |
AJXRZKIHWZAXJZ
|
6.9 | IC50 | 3 | — | |
IBKWYNPFFOZRLP
|
6.9 | IC50 | 4 | — | |
BBDSYVIXESVDPE
|
6.9 | IC50 | 4 | — | |
DIDJYPFYHDBXHU
|
6.9 | IC50 | 4 | — | |
FTWCGCABDYPPKS
|
6.9 | IC50 | 4 | — | |
QRIXKWMQRHCONV
|
6.9 | IC50 | 4 | — | |
SDVAHCXGDGYWFA
|
6.9 | IC50 | 12 | — | |
WNEODWDFDXWOLU
|
6.9 | Kd | 5 | — | |
LSJWYMSFUWBGPN
|
6.9 | IC50 | 17 | — | |
VXJXHNMYRAHBBO
|
6.9 | IC50 | 5 | — | |
CEUSZLVORFRBCV
|
6.8 | IC50 | 13 | — | |
UBUVIQYWARUKMQ
|
6.8 | IC50 | 4 | — | |
YHNFAXONRPKPAO
|
6.8 | IC50 | 2 | — | |
DPRNXTSMYVCYLJ
|
6.8 | IC50 | 13 | — | |
GEEUDEOZMWBPDT
|
6.8 | IC50 | 4 | — | |
LUMAVJBHSUJPOG
|
6.8 | IC50 | 4 | — | |
HKSZLNNOFSGOKW
|
6.8 | Kd | 408 | — | |
HKSZLNNOFSGOKW
|
6.8 | Kd | 213 | — | |
FHOKFOHRQUSPMF
|
6.8 | IC50 | 3 | — | |
KJRVCMVPIKELBC
|
6.8 | IC50 | 12 | — | |
MUSDVFBSNCGDJV
|
6.8 | IC50 | 3 | — | |
FNNWNXFWBPLQIV
|
6.7 | IC50 | 3 | — | |
NHHQJBCNYHBUSI
|
6.7 | Kd | 220 | — | |
OMZCMEYTWSXEPZ
|
6.7 | IC50 | 43 | Yes | |
UMBDWDIRLTVPBF
|
6.7 | IC50 | 9 | — | |
CXQHYVUVSFXTMY
|
6.7 | Kd | 154 | — | |
GZYUJXFTHLKPAK
|
6.7 | IC50 | 16 | — | |
PBLPUMCTPXMGKZ
|
6.7 | IC50 | 2 | — | |
SEJGTFPOEJWEGG
|
6.7 | Kd | 149 | — | |
TXIUPNHPXDVAAM
|
6.7 | IC50 | 5 | — | |
UIARLYUEJFELEN
|
6.7 | Kd | 289 | Yes | |
WVXNSAVVKYZVOE
|
6.7 | IC50 | 92 | — | |
RKUNGXOSUGLQJY
|
6.7 | IC50 | 3 | — | |
JJORFRRMKVGMOJ
|
6.6 | IC50 | 3 | — | |
PUIXMSRTTHLNKI
|
6.6 | IC50 | 12 | — | |
UEFCSGDOOJJXTN
|
6.6 | IC50 | 46 | — | |
GKZGJDDKZTVQJZ
|
6.5 | IC50 | 4 | — | |
NFLKTKKJFVNGLH
|
6.5 | IC50 | 4 | — | |
VQUUBQYYHFHNFA
|
6.5 | IC50 | 4 | — | |
HTUBKQUPEREOGA
|
6.5 | IC50 | 6 | Yes | |
LAUHLGUSVSJYCI
|
6.5 | IC50 | 16 | — | |
UQDKCJOIUBVSRC
|
6.5 | IC50 | 2 | — | |
VVPLAYNPERQXNL
|
6.5 | IC50 | 3 | — | |
GLBZSOQDAOLMGC
|
6.4 | IC50 | 23 | Yes |