Target Details
| UniProt AC | P51813 |
|---|---|
| Gene Symbol | BMX |
| Protein Name | Cytoplasmic tyrosine-protein kinase BMX |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00779 (BTK) PF00169 (PH) PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) |
Summary
- Multi-target molecules 226
- Clinical molecules 11
- Avg pChEMBL 7.47
Active Molecules (226)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DNDCQFCAXLONFM
|
7.6 | IC50 | 4 | — | |
KQISOZQPFQHIFH
|
7.6 | IC50 | 4 | — | |
WCCLANJGOUJNNL
|
7.6 | IC50 | 4 | — | |
CEJHRMYKGWBHHX
|
7.6 | IC50 | 3 | — | |
MHGMKTVDZXADNH
|
7.6 | IC50 | 4 | — | |
AHBFBRPGNOVEBK
|
7.5 | IC50 | 11 | — | |
LCJSUUXDTVNFHO
|
7.5 | IC50 | 3 | — | |
SXLIACXIXLLKGR
|
7.5 | IC50 | 4 | — | |
VAARYSWULJUGST
|
7.5 | Kd | 119 | Yes | |
ZRYMMWAJAFUANM
|
7.5 | IC50 | 7 | — | |
ZZJOFPXLPFXEKV
|
7.5 | IC50 | 4 | — | |
ZXGCNNKDPNECIS
|
7.5 | IC50 | 4 | — | |
DOVHWPFJHQGYDS
|
7.5 | IC50 | 4 | — | |
HGXKBKYPMMTKKK
|
7.5 | IC50 | 3 | — | |
LJBPJECYFQWDEL
|
7.5 | IC50 | 3 | — | |
QUIWHXQETADMGN
|
7.5 | IC50 | 4 | — | |
IGXJXMLDIIGDNE
|
7.4 | IC50 | 8 | — | |
IRMJEKARXQRXOY
|
7.4 | IC50 | 3 | — | |
OSAWFUCUZJNEID
|
7.4 | IC50 | 20 | — | |
PTHVKCSYXICMAR
|
7.4 | IC50 | 14 | — | |
SFCBIFOAGRZJNX
|
7.4 | Kd | 22 | — | |
DNFWTELNLRENAM
|
7.4 | IC50 | 4 | — | |
NMNLVTJEQAQJHN
|
7.4 | IC50 | 4 | — | |
RJARQSDFMBQVEH
|
7.4 | IC50 | 4 | — | |
FWTHOUYYKYVNTG
|
7.4 | IC50 | 2 | — | |
ISQNGOQQSMUJCK
|
7.4 | IC50 | 3 | — | |
CVBABGVEYUMHNU
|
7.3 | IC50 | 6 | — | |
HDVYJNSAOAUAIQ
|
7.3 | IC50 | 4 | — | |
WDENQIQQYWYTPO
|
7.3 | IC50 | 8 | — | |
JNXAHUQUDHQPOY
|
7.3 | IC50 | 3 | — | |
OKKLVTXFDLVHSC
|
7.3 | IC50 | 2 | — | |
ITTRLTNMFYIYPA
|
7.3 | IC50 | 17 | — | |
KRILZVCKKUOPKH
|
7.3 | IC50 | 4 | — | |
UORAPQCBWYIISR
|
7.3 | IC50 | 15 | — | |
WZLCFQWCRHXUJG
|
7.3 | IC50 | 4 | — | |
KOQJXUXLQGQJDF
|
7.2 | IC50 | 4 | — | |
RMTJSBZCZKCYHB
|
7.2 | IC50 | 13 | — | |
ZTUJNJAKTLHBEX
|
7.2 | IC50 | 5 | — | |
WMMNTQFZCHUZSM
|
7.2 | IC50 | 14 | — | |
YYRYNQBAVOOSOA
|
7.2 | IC50 | 4 | — | |
ZFKUIXUALOAFLP
|
7.2 | IC50 | 3 | — | |
GUGCOQNZIOTJQQ
|
7.1 | IC50 | 3 | — | |
ZYQIUDPJBOUHCC
|
7.1 | IC50 | 4 | — | |
LXURGGKEOPHREO
|
7.1 | IC50 | 13 | — | |
PENAJAQLAALQQB
|
7.1 | IC50 | 3 | — | |
SVIHDEUPJUWZRH
|
7.1 | IC50 | 2 | — | |
VTJHGMZHVOXJPG
|
7.1 | IC50 | 15 | — | |
BLOSAGLLXHJECN
|
7.1 | IC50 | 4 | — | |
JSAQBOQCZJHWMA
|
7.1 | Kd | 11 | — | |
OPKHZFMFWCMAPS
|
7.0 | IC50 | 6 | — |