Target Details
| UniProt AC | P51813 |
|---|---|
| Gene Symbol | BMX |
| Protein Name | Cytoplasmic tyrosine-protein kinase BMX |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00779 (BTK) PF00169 (PH) PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) |
Summary
- Multi-target molecules 226
- Clinical molecules 11
- Avg pChEMBL 7.47
Active Molecules (226)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UBPYILGKFZZVDX
|
8.1 | IC50 | 130 | Yes | |
UVUTZINLTAEGAD
|
8.1 | IC50 | 4 | — | |
VUDJPBPVCUEFHU
|
8.1 | IC50 | 5 | — | |
KWYIQYSIXKBGBV
|
8.1 | IC50 | 2 | — | |
LJODJUIHONTDMR
|
8.1 | IC50 | 7 | — | |
ILXFYIOJPFUYGX
|
8.1 | IC50 | 5 | — | |
NZIQNLGMMJGSQU
|
8.0 | IC50 | 6 | — | |
XNPHXLCYBBQUQK
|
8.0 | IC50 | 4 | — | |
COWVAFPFSREMEQ
|
8.0 | IC50 | 5 | — | |
DBNDRMANPSPBJX
|
8.0 | IC50 | 3 | — | |
FMRJPPUXBYSJRE
|
8.0 | IC50 | 4 | — | |
JUSWPUDQOKINJO
|
8.0 | IC50 | 16 | — | |
SRSQULBCTWSVKL
|
8.0 | IC50 | 15 | — | |
VREZKFPACUPTJS
|
8.0 | IC50 | 5 | — | |
XURALSVDCFXBAX
|
8.0 | IC50 | 4 | — | |
CDFHNEWIEMNZKE
|
7.9 | IC50 | 4 | — | |
KOIOINMFIPQGKH
|
7.9 | IC50 | 3 | — | |
KPZGJWPPVXZLDN
|
7.9 | IC50 | 10 | — | |
CDISOBGWDHAHGF
|
7.9 | IC50 | 16 | — | |
GFHLXZJWIUHXCL
|
7.9 | IC50 | 5 | — | |
GFZZUAFZBKEOHV
|
7.9 | IC50 | 7 | — | |
GXANJKDFGYJBEM
|
7.9 | IC50 | 5 | — | |
SLKAFUZHONQYQY
|
7.9 | IC50 | 5 | — | |
MZSDTUIZKGUVHK
|
7.8 | IC50 | 4 | — | |
SBRIQINKAOKMMM
|
7.8 | IC50 | 6 | — | |
SEJLPXCPMNSRAM
|
7.8 | IC50 | 7 | — | |
YGPHJRJCXOYFAN
|
7.8 | IC50 | 3 | — | |
VOUOPUKEZYZDGH
|
7.8 | IC50 | 3 | — | |
XIDJFSRGLOUDGG
|
7.8 | IC50 | 4 | — | |
XZAATUBTUPPERZ
|
7.8 | IC50 | 6 | — | |
ZFDGMDVYMNWICG
|
7.8 | IC50 | 10 | — | |
JGLBGBDMKMGQFA
|
7.8 | IC50 | 5 | — | |
OXOMWFOJARKFIY
|
7.8 | IC50 | 4 | — | |
SXXRMKLCTXMFPH
|
7.8 | IC50 | 5 | — | |
CLKNHJDZJCCLAZ
|
7.8 | IC50 | 4 | — | |
SVLLKLFGGWAXTK
|
7.8 | IC50 | 5 | — | |
JXVBUPCEADJXCV
|
7.7 | IC50 | 4 | — | |
LQSGDXCDNZWTJN
|
7.7 | IC50 | 17 | — | |
OMIQRSKHABIPRH
|
7.7 | IC50 | 15 | — | |
YTIWDAUDJMCXOD
|
7.7 | IC50 | 5 | — | |
LVQAGIXEFVAFEO
|
7.7 | IC50 | 2 | — | |
FJNULDLUBJRUJN
|
7.7 | IC50 | 5 | — | |
OPHSZSZDICRBPP
|
7.7 | IC50 | 16 | — | |
XYFZVVYVIFJBIS
|
7.7 | IC50 | 17 | — | |
ATLOUNJJIAISOI
|
7.7 | IC50 | 4 | — | |
SIFFAYSEHIUEHK
|
7.7 | IC50 | 4 | — | |
YHVHYWYQEFELOW
|
7.7 | IC50 | 44 | — | |
VRCBGBBYFHLJRE
|
7.7 | IC50 | 5 | — | |
QNNJMWIVIVLSHC
|
7.6 | IC50 | 4 | — | |
TVJRDCQUZMGBAB
|
7.6 | IC50 | 13 | — |