Target Details
UniProt ACP51813
Gene SymbolBMX
Protein NameCytoplasmic tyrosine-protein kinase BMX
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00779 (BTK) PF00169 (PH) PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2)
Summary
  • Multi-target molecules 226
  • Clinical molecules 11
  • Avg pChEMBL 7.47
Top Co-occurrence Targets
Active Molecules (226)
InChIKey pChEMBL Type Targets Clinical
XYFPWWZEPKGCCK 9.4 IC50 7
IZLUBQPWEKVIDI 9.4 IC50 5
NNGVMERLTTVLQP 9.2 IC50 8
SMOPKEHQPPXRSH 9.2 IC50 8
LCYSSHSIKSARGO 9.1 IC50 19
XYFPWWZEPKGCCK 9.1 IC50 34
XYFPWWZEPKGCCK 9.1 IC50 7
SQFDBQCBXUWICP 9.1 IC50 3
LCFFREMLXLZNHE 9.0 IC50 5
SSDFTYWIYVWCIE 9.0 IC50 17
AXEVKNAHSSENFT 8.9 IC50 5
BJMXICGJKUALLN 8.9 IC50 8
HJAUUHMYFPHMCT 8.9 IC50 4
PZWSKESWDIFAFK 8.8 IC50 9
ZBNZXTGUTAYRHI 8.8 Kd 102 Yes
ZWVLMQTXUWMUII 8.8 IC50 9 Yes
YMSXHRWUGLAAKL 8.8 IC50 14 Yes
WZLQKELQHIYATN 8.8 IC50 4
KZMQPYCXSAGLTB 8.7 IC50 8
PWISMKGZBHMEFG 8.7 IC50 6
RZSSIBVYFFJHNU 8.7 IC50 4
VKQPGLDQSGLMMO 8.6 IC50 4
CMFVTAHMZDUCJB 8.6 IC50 10
MQSCGRDOQBVIMP 8.6 IC50 5
BUNVZNMOFRWGMI 8.5 IC50 6
NGZPCPROZUYFJJ 8.5 IC50 6
XXJWOZLYIDMCJH 8.5 IC50 4
LHFAKDSSXLAPAE 8.5 IC50 4
KXBDTLQSDKGAEB 8.5 IC50 8
GOOMNGHXGYAHJM 8.5 IC50 7
AOKKWYGSIRAXIZ 8.5 IC50 4
LYADGAGFYYXXIO 8.5 IC50 82
VYZQSAKXLMEDCB 8.4 IC50 9
DJKOMFSZAABEBE 8.4 IC50 4
DQFOPMWZUFUHDC 8.3 IC50 6
QCJFYACTZIVZBB 8.3 IC50 8
RNOAOAWBMHREKO 8.3 IC50 15
BZWACBLCIHAEKY 8.2 IC50 5
FUZSHLVNKZZEKR 8.2 IC50 16
VJPPLCNBDLZIFG 8.2 IC50 5
XNVVTSSPSNFSCT 8.2 IC50 3
BNRXMSGHPVYSDK 8.2 IC50 24
BTWVWABAWDKQNJ 8.2 IC50 8
RTRNJQOBEOISFQ 8.2 IC50 5
IRBVGTPPFBYDKX 8.2 IC50 9
JMVDIGHUQAXWIE 8.1 IC50 10
SXXABOHFQFARBT 8.1 IC50 5
MNDLPZPZVIEBFF 8.1 IC50 4
SFMJNHNUOVADRW 8.1 IC50 7
SZNYUUZOQHNEKB 8.1 IC50 7
2D structure