Target Details
| UniProt AC | P51813 |
|---|---|
| Gene Symbol | BMX |
| Protein Name | Cytoplasmic tyrosine-protein kinase BMX |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00779 (BTK) PF00169 (PH) PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) |
Summary
- Multi-target molecules 226
- Clinical molecules 11
- Avg pChEMBL 7.47
Active Molecules (226)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XYFPWWZEPKGCCK
|
9.4 | IC50 | 7 | — | |
IZLUBQPWEKVIDI
|
9.4 | IC50 | 5 | — | |
NNGVMERLTTVLQP
|
9.2 | IC50 | 8 | — | |
SMOPKEHQPPXRSH
|
9.2 | IC50 | 8 | — | |
LCYSSHSIKSARGO
|
9.1 | IC50 | 19 | — | |
XYFPWWZEPKGCCK
|
9.1 | IC50 | 34 | — | |
XYFPWWZEPKGCCK
|
9.1 | IC50 | 7 | — | |
SQFDBQCBXUWICP
|
9.1 | IC50 | 3 | — | |
LCFFREMLXLZNHE
|
9.0 | IC50 | 5 | — | |
SSDFTYWIYVWCIE
|
9.0 | IC50 | 17 | — | |
AXEVKNAHSSENFT
|
8.9 | IC50 | 5 | — | |
BJMXICGJKUALLN
|
8.9 | IC50 | 8 | — | |
HJAUUHMYFPHMCT
|
8.9 | IC50 | 4 | — | |
PZWSKESWDIFAFK
|
8.8 | IC50 | 9 | — | |
ZBNZXTGUTAYRHI
|
8.8 | Kd | 102 | Yes | |
ZWVLMQTXUWMUII
|
8.8 | IC50 | 9 | Yes | |
YMSXHRWUGLAAKL
|
8.8 | IC50 | 14 | Yes | |
WZLQKELQHIYATN
|
8.8 | IC50 | 4 | — | |
KZMQPYCXSAGLTB
|
8.7 | IC50 | 8 | — | |
PWISMKGZBHMEFG
|
8.7 | IC50 | 6 | — | |
RZSSIBVYFFJHNU
|
8.7 | IC50 | 4 | — | |
VKQPGLDQSGLMMO
|
8.6 | IC50 | 4 | — | |
CMFVTAHMZDUCJB
|
8.6 | IC50 | 10 | — | |
MQSCGRDOQBVIMP
|
8.6 | IC50 | 5 | — | |
BUNVZNMOFRWGMI
|
8.5 | IC50 | 6 | — | |
NGZPCPROZUYFJJ
|
8.5 | IC50 | 6 | — | |
XXJWOZLYIDMCJH
|
8.5 | IC50 | 4 | — | |
LHFAKDSSXLAPAE
|
8.5 | IC50 | 4 | — | |
KXBDTLQSDKGAEB
|
8.5 | IC50 | 8 | — | |
GOOMNGHXGYAHJM
|
8.5 | IC50 | 7 | — | |
AOKKWYGSIRAXIZ
|
8.5 | IC50 | 4 | — | |
LYADGAGFYYXXIO
|
8.5 | IC50 | 82 | — | |
VYZQSAKXLMEDCB
|
8.4 | IC50 | 9 | — | |
DJKOMFSZAABEBE
|
8.4 | IC50 | 4 | — | |
DQFOPMWZUFUHDC
|
8.3 | IC50 | 6 | — | |
QCJFYACTZIVZBB
|
8.3 | IC50 | 8 | — | |
RNOAOAWBMHREKO
|
8.3 | IC50 | 15 | — | |
BZWACBLCIHAEKY
|
8.2 | IC50 | 5 | — | |
FUZSHLVNKZZEKR
|
8.2 | IC50 | 16 | — | |
VJPPLCNBDLZIFG
|
8.2 | IC50 | 5 | — | |
XNVVTSSPSNFSCT
|
8.2 | IC50 | 3 | — | |
BNRXMSGHPVYSDK
|
8.2 | IC50 | 24 | — | |
BTWVWABAWDKQNJ
|
8.2 | IC50 | 8 | — | |
RTRNJQOBEOISFQ
|
8.2 | IC50 | 5 | — | |
IRBVGTPPFBYDKX
|
8.2 | IC50 | 9 | — | |
JMVDIGHUQAXWIE
|
8.1 | IC50 | 10 | — | |
SXXABOHFQFARBT
|
8.1 | IC50 | 5 | — | |
MNDLPZPZVIEBFF
|
8.1 | IC50 | 4 | — | |
SFMJNHNUOVADRW
|
8.1 | IC50 | 7 | — | |
SZNYUUZOQHNEKB
|
8.1 | IC50 | 7 | — |