Target Details
| UniProt AC | P51812 |
|---|---|
| Gene Symbol | RPS6KA3 |
| Protein Name | Ribosomal protein S6 kinase alpha-3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 322
- Clinical molecules 28
- Avg pChEMBL 6.85
KEGG Pathways (10)
Associated Diseases (2)
Active Molecules (322)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MMWVUKRVNHSCOU
|
6.0 | IC50 | 2 | — | |
AWJPVXSHMIELNJ
|
6.0 | Ki | 23 | — | |
BIIVYFLTOXDAOV
|
6.0 | Kd | 82 | Yes | |
BPNUQXPIQBZCMR
|
6.0 | Ki | 60 | — | |
HOBMVEVXDIOMDM
|
6.0 | Ki | 18 | — | |
IMLXFZLHOPEBPM
|
6.0 | Ki | 12 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
JBRASADWXDKCLJ
|
6.0 | Ki | 22 | — | |
JVUYFKGAACUDSV
|
6.0 | IC50 | 2 | — | |
KDKUVYLMPJIGKA
|
6.0 | Ki | 91 | Yes | |
LCKDESRGCHSHHO
|
6.0 | Ki | 18 | — | |
LRZYYIZFBXFSJB
|
6.0 | Ki | 69 | — | |
MASJMHFQMYAPJR
|
6.0 | Ki | 41 | — | |
NGOGFTYYXHNFQH
|
6.0 | Ki | 15 | — | |
PCQMERRARZKTPW
|
6.0 | Ki | 68 | — | |
PFCUZXCHLYIMTJ
|
6.0 | Ki | 18 | — | |
QJIVDCJIPGAKQZ
|
6.0 | Ki | 25 | — | |
RWEHAHIEUDLKGT
|
6.0 | Ki | 33 | — | |
UIRCQOKSJDLYBB
|
6.0 | Ki | 50 | — | |
XDOILUADECHLAS
|
6.0 | IC50 | 2 | — | |
YXUQWISLOFXNGN
|
6.0 | Ki | 16 | — | |
YYPKOMNJRZRWIC
|
6.0 | Ki | 26 | — |