Target Details
| UniProt AC | P51812 |
|---|---|
| Gene Symbol | RPS6KA3 |
| Protein Name | Ribosomal protein S6 kinase alpha-3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 322
- Clinical molecules 28
- Avg pChEMBL 6.85
KEGG Pathways (10)
Associated Diseases (2)
Active Molecules (322)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SEZFNTZQMWJIAI
|
6.2 | Ki | 22 | — | |
SFPWNTQWFFNJIH
|
6.2 | Ki | 48 | — | |
WHVFDYQCAMPLMS
|
6.2 | Ki | 20 | Yes | |
WPHKIQPVPYJNAX
|
6.2 | Ki | 81 | — | |
YMIJUBCSOKSFRU
|
6.2 | Ki | 87 | — | |
ZGDYBJXDIXVTLV
|
6.2 | Ki | 54 | — | |
FKMYIGXYIAVMND
|
6.2 | IC50 | 3 | — | |
MJSXSLBYCSPRHR
|
6.2 | IC50 | 10 | Yes | |
QCPXWEFKAZRXTO
|
6.2 | IC50 | 3 | — | |
OBYOBQZFZXGFMP
|
6.2 | IC50 | 3 | — | |
XLFNLJYGUOLEJS
|
6.2 | IC50 | 26 | — | |
FMGZGKDQXIZQLF
|
6.1 | IC50 | 2 | — | |
BMGQWWVMWDBQGC
|
6.1 | Kd | 147 | Yes | |
FLBNLJLONKAPLR
|
6.1 | Kd | 31 | — | |
UQVVQLRAEQBLIK
|
6.1 | IC50 | 2 | — | |
AHJRHEGDXFFMBM
|
6.1 | Ki | 28 | — | |
AUDNGNGLLRZLDR
|
6.1 | Ki | 33 | — | |
DPRGOXVMSNDADU
|
6.1 | Ki | 16 | — | |
DZIPQNPWTUXXSJ
|
6.1 | Ki | 18 | — | |
DZSUJUOJJJCWGG
|
6.1 | Ki | 55 | Yes | |
GHMRUNOHAHJNNA
|
6.1 | Ki | 29 | — | |
HEUSUIRCBWROMH
|
6.1 | Ki | 64 | — | |
JNXJKTXDSPWNRP
|
6.1 | Ki | 30 | — | |
LKUJDAHYLPICSE
|
6.1 | Ki | 24 | — | |
MHWHPWMWKYXCRJ
|
6.1 | Ki | 32 | — | |
MJMWZFLAXXUPEE
|
6.1 | Ki | 2 | — | |
NKEUPUJTVALZIK
|
6.1 | Ki | 28 | — | |
NWBMEZSCKMLUTH
|
6.1 | IC50 | 3 | — | |
NZVDDFRUBIEKLV
|
6.1 | Ki | 20 | — | |
OPLHMHMCXQXEQG
|
6.1 | Ki | 10 | — | |
ORRHVRJUSPCILV
|
6.1 | Ki | 16 | — | |
PJUVRETYCLPAFV
|
6.1 | Ki | 20 | — | |
QVNZKVACBBTKSL
|
6.1 | Ki | 38 | — | |
RITAVMQDGBJQJZ
|
6.1 | Ki | 33 | — | |
SBFPHSVZEXSHTL
|
6.1 | Ki | 62 | — | |
SGHXFHRRWFLILP
|
6.1 | Ki | 29 | — | |
TVEREFRWBLRPPJ
|
6.1 | Ki | 15 | — | |
URNZTLZSAVLTIZ
|
6.1 | Ki | 26 | — | |
UXUQVXDYXKMCGA
|
6.1 | Ki | 21 | — | |
UYGYYOIUVFMGKQ
|
6.1 | Ki | 30 | — | |
VCFDMLBPASGZTP
|
6.1 | Ki | 38 | — | |
WUBHCQHBUVGGRX
|
6.1 | Ki | 11 | — | |
XHORJSJFHVABEA
|
6.1 | Ki | 49 | — | |
XOOAAYRIVATZNM
|
6.1 | Ki | 55 | — | |
ZLHFILGSQDJULK
|
6.1 | Ki | 37 | Yes | |
PROGKLMIRQVLRO
|
6.1 | IC50 | 12 | — | |
QKVFMAAIXZONRN
|
6.0 | IC50 | 2 | — | |
HWTKDUIKACSTLX
|
6.0 | IC50 | 2 | — | |
JXFASNVVYCKOKY
|
6.0 | IC50 | 2 | — | |
KCVOKHWVSRPHJC
|
6.0 | IC50 | 2 | — |