Target Details
| UniProt AC | P51812 |
|---|---|
| Gene Symbol | RPS6KA3 |
| Protein Name | Ribosomal protein S6 kinase alpha-3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 322
- Clinical molecules 28
- Avg pChEMBL 6.85
KEGG Pathways (10)
Associated Diseases (2)
Active Molecules (322)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NECQZMQPXFYVOY
|
6.7 | Ki | 26 | — | |
PYXQMJSGJIJHJT
|
6.7 | Ki | 28 | — | |
SUULIUKTZNKMMB
|
6.7 | Ki | 10 | — | |
UVZVWLFSZNPMBS
|
6.7 | Ki | 17 | — | |
VKBFHTIUXUCYRQ
|
6.7 | Ki | 66 | — | |
VNGYQBMDQMDALH
|
6.7 | Ki | 25 | — | |
YEHCNYAQEBQCCS
|
6.7 | Ki | 74 | — | |
CHFKZEPYDHGBQK
|
6.7 | IC50 | 2 | — | |
WGAAHZPAINDSDB
|
6.7 | IC50 | 2 | — | |
AATRJMCVLUZFSH
|
6.7 | IC50 | 2 | — | |
FLSKMXCIDGMHDI
|
6.7 | IC50 | 2 | — | |
LHRDCIRKYUFYOY
|
6.7 | IC50 | 2 | — | |
DUGXSNHFGBPCPM
|
6.6 | IC50 | 2 | — | |
GPNUVUGMFDKAJH
|
6.6 | IC50 | 4 | — | |
GSXRCPJTNIGKSZ
|
6.6 | Ki | 43 | — | |
JXMYIDZREHNPDO
|
6.6 | Ki | 19 | — | |
LGHBDVLAHHANMX
|
6.6 | Ki | 53 | — | |
MQRDVGBWWVWMEN
|
6.6 | Ki | 47 | — | |
NHFDRBXTEDBWCZ
|
6.6 | Ki | 41 | — | |
PTVPBWWDGZSEAF
|
6.6 | Ki | 63 | — | |
UDFDIIVNIYWXDM
|
6.6 | Ki | 74 | — | |
XLFYOIVELARSKP
|
6.6 | Ki | 33 | — | |
YARFNYLGLQVPEB
|
6.6 | IC50 | 2 | — | |
NNQHKTWARZSGTQ
|
6.6 | IC50 | 7 | — | |
QNABDSWBQJKBHK
|
6.6 | IC50 | 45 | — | |
BTCGJYJHCYOBJS
|
6.6 | IC50 | 2 | — | |
YYLKKYCXAOBSRM
|
6.5 | Kd | 191 | — | |
NMSKCMQPIFOSHU
|
6.5 | IC50 | 2 | — | |
UIARLYUEJFELEN
|
6.5 | Kd | 289 | Yes | |
JYYLVUFNAHSSFE
|
6.5 | Kd | 9 | — | |
DPEXRCOBPACFOO
|
6.5 | Ki | 36 | — | |
KJVWCDAPVMWKLJ
|
6.5 | Ki | 20 | — | |
PDBPUXLUVDSLML
|
6.5 | Ki | 14 | — | |
PIQCTGMSNWUMAF
|
6.5 | Ki | 137 | Yes | |
PNKALLUVKOKYHZ
|
6.5 | Ki | 32 | — | |
QAJPIJHWTGPUNZ
|
6.5 | Ki | 37 | — | |
SKLNUYVBOFIJAT
|
6.5 | Ki | 5 | — | |
USHMNZBDAOGLMB
|
6.5 | Ki | 26 | — | |
VGNKOJURPOHWJF
|
6.5 | Ki | 21 | — | |
VSVWQTDDGQSGHP
|
6.5 | Ki | 51 | — | |
QBWKPGNFQQJGFY
|
6.5 | IC50 | 5 | Yes | |
OTMPGQSHVZZPJK
|
6.5 | IC50 | 2 | — | |
SKDSRJRRAQLUPP
|
6.4 | IC50 | 8 | Yes | |
XEMRFXZAJHTFCF
|
6.4 | IC50 | 2 | — | |
YBYYWUUUGCNAHQ
|
6.4 | IC50 | 8 | — | |
SXOZSDJHGMAEGZ
|
6.4 | IC50 | 2 | — | |
UEFCSGDOOJJXTN
|
6.4 | IC50 | 46 | — | |
ACNCCUVYXQGPKZ
|
6.4 | Ki | 31 | — | |
AOFJRBMLTUGMMP
|
6.4 | Ki | 12 | — | |
CLRFYTGANQZOBS
|
6.4 | Ki | 41 | — |