Target Details
| UniProt AC | P51812 |
|---|---|
| Gene Symbol | RPS6KA3 |
| Protein Name | Ribosomal protein S6 kinase alpha-3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 322
- Clinical molecules 28
- Avg pChEMBL 6.85
KEGG Pathways (10)
Associated Diseases (2)
Active Molecules (322)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UJBJWYNPUOLFIZ
|
7.1 | IC50 | 49 | — | |
AXRCEOKUDYDWLF
|
7.1 | Kd | 31 | — | |
LQZKYXLZCLMOGP
|
7.1 | IC50 | 2 | — | |
VSYFECVWSJTEIL
|
7.1 | IC50 | 2 | — | |
CPDJVFPDCVMFHF
|
7.0 | IC50 | 2 | — | |
PXRIUZVVLPVSSH
|
7.0 | IC50 | 2 | — | |
FUMCKNCUEAQHCV
|
7.0 | Ki | 103 | — | |
HIUHVDROHDSKTC
|
7.0 | Ki | 20 | — | |
JJGSOVIZOMZMCS
|
7.0 | Ki | 35 | — | |
NJKBCVHYFWYIIQ
|
7.0 | Ki | 2 | — | |
NKGLJTITEFZKAN
|
7.0 | Ki | 35 | — | |
PROLIXHVRCJEFH
|
7.0 | Ki | 46 | — | |
TVUWQDLBEOZVOU
|
7.0 | Ki | 41 | — | |
XPHWIERLJBFPFV
|
7.0 | Ki | 69 | — | |
QDIMOURDMVMOHZ
|
7.0 | IC50 | 3 | — | |
MVRDTJDXYOJXNF
|
7.0 | IC50 | 2 | — | |
JBOKTWNEIMBJNQ
|
7.0 | IC50 | 2 | — | |
UTARVXNWFXWXPH
|
7.0 | IC50 | 2 | — | |
YVQOYBIBWBAHKH
|
6.9 | IC50 | 12 | — | |
DKSNLQYRZJKYOC
|
6.9 | Ki | 51 | — | |
DTMZXHDQZQLTHA
|
6.9 | Ki | 21 | — | |
JCFJQIHDZHHMQT
|
6.9 | Ki | 42 | — | |
OAVGBZOFDPFGPJ
|
6.9 | Ki | 42 | Yes | |
RGNHKJWHFIPHIM
|
6.9 | Ki | 66 | — | |
TUJUZVJICDSNLY
|
6.9 | Ki | 19 | — | |
XCHWBXBDZRJVDP
|
6.9 | Ki | 51 | — | |
FTOWCRNOCYACIS
|
6.8 | IC50 | 2 | — | |
KKKRKRMVJRHDMG
|
6.8 | Kd | 14 | — | |
CFIBXVQLBVNOHW
|
6.8 | Ki | 64 | — | |
KKYPRNBBPBRJQX
|
6.8 | Ki | 40 | — | |
LHQWPYOYDRVMFI
|
6.8 | Ki | 21 | — | |
SHENEEFOURUIBP
|
6.8 | Ki | 29 | — | |
TWZVBMXTDSNZLS
|
6.8 | Ki | 7 | — | |
UOVCGJXDGOGOCZ
|
6.8 | Ki | 59 | — | |
WUWDLXZGHZSWQZ
|
6.8 | Ki | 41 | — | |
XZWVOUQIYLZUCJ
|
6.8 | Ki | 23 | — | |
ZKHDDJKHTPLPOQ
|
6.8 | Ki | 62 | — | |
ZVPDNRVYHLRXLX
|
6.8 | Ki | 35 | Yes | |
DKZYXHCYPUVGAF
|
6.8 | Kd | 112 | — | |
HZTYDQRUAWIZRE
|
6.8 | Kd | 40 | Yes | |
UERCXNOQFSTSOY
|
6.8 | IC50 | 2 | — | |
GMVUXANRAYNFHC
|
6.7 | IC50 | 2 | — | |
RHAMYMXUVZEEJR
|
6.7 | IC50 | 4 | — | |
RHGZQGXELRMGES
|
6.7 | IC50 | 8 | Yes | |
WINHZLLDWRZWRT
|
6.7 | Kd | 201 | Yes | |
WXEZWMNXEPCNCY
|
6.7 | IC50 | 2 | — | |
ZHJGWYRLJUCMRT
|
6.7 | Kd | 18 | — | |
GCBJDOWIQHMCMR
|
6.7 | Ki | 84 | — | |
IPKHSYHXXAIZDD
|
6.7 | Ki | 18 | — | |
MFAQYJIYDMLAIM
|
6.7 | Kd | 130 | Yes |