Target Details
| UniProt AC | P51812 |
|---|---|
| Gene Symbol | RPS6KA3 |
| Protein Name | Ribosomal protein S6 kinase alpha-3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 322
- Clinical molecules 28
- Avg pChEMBL 6.85
KEGG Pathways (10)
Associated Diseases (2)
Active Molecules (322)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QYLAYPRSSJNQDC
|
7.7 | IC50 | 2 | — | |
VCZQSUBZCZZLAX
|
7.7 | IC50 | 2 | — | |
XRTXYXCNVWUOKB
|
7.7 | IC50 | 2 | — | |
ZCBUQCWBWNUWSU
|
7.7 | Ki | 11 | — | |
ZDYXRELDNKSUBF
|
7.7 | IC50 | 2 | — | |
KAKNBLVUBRXYQD
|
7.7 | IC50 | 2 | — | |
AYCPARAPKDAOEN
|
7.7 | IC50 | 73 | — | |
DTEKTGDVSARYDS
|
7.6 | IC50 | 11 | — | |
BTHYNSZFAHGSOX
|
7.6 | IC50 | 4 | — | |
GWJHMRBQEUHFOC
|
7.6 | Ki | 42 | — | |
MVJMMLFMPWITEJ
|
7.6 | Ki | 110 | — | |
QTQUAHGXBLFSCH
|
7.6 | Ki | 10 | — | |
AILRADAXUVEEIR
|
7.6 | IC50 | 75 | — | |
XLYVQVWMTOLDNL
|
7.5 | IC50 | 21 | — | |
XLYVQVWMTOLDNL
|
7.5 | IC50 | 21 | — | |
YVUHNKZPGGBYDH
|
7.5 | IC50 | 2 | — | |
RSFBRAHCHZGZPB
|
7.5 | IC50 | 8 | — | |
SDBOIBYRBWPIEL
|
7.5 | Ki | 31 | — | |
ZHMXXVNQAFCXKK
|
7.4 | IC50 | 2 | — | |
GCYXEGSPUDSZJY
|
7.4 | Ki | 82 | — | |
HWXDZAYQHRBBQT
|
7.4 | IC50 | 2 | — | |
LOCWELCIOZHZHE
|
7.4 | Ki | 11 | — | |
PHWHNHYZZNJPLB
|
7.4 | Ki | 16 | — | |
YOVNFNXUCOWYSG
|
7.4 | Ki | 33 | Yes | |
ZQMGSEHFOOINGT
|
7.4 | IC50 | 2 | — | |
WIICYVHPNFINMO
|
7.4 | IC50 | 2 | — | |
ULNZFQKAFXCYBO
|
7.4 | IC50 | 2 | — | |
NGFGTMFVWSDFPS
|
7.3 | IC50 | 32 | — | |
ZVYLAQPDMUKXOT
|
7.3 | IC50 | 5 | — | |
FLEAYYMORDPWAJ
|
7.3 | Ki | 90 | — | |
LCVZRKFDNWPBET
|
7.3 | IC50 | 2 | — | |
RKUKAACYUCUJEE
|
7.3 | Ki | 58 | — | |
WAKGEHXTOOFEAE
|
7.3 | Ki | 27 | — | |
ZHRYDDVDLCQYQA
|
7.3 | Ki | 5 | — | |
LZAHKCVOJMJNFW
|
7.3 | IC50 | 2 | — | |
OZFFKOSQNBBYCA
|
7.3 | IC50 | 12 | — | |
ZWUCWBYYVLQXEP
|
7.2 | IC50 | 4 | — | |
HKSZLNNOFSGOKW
|
7.2 | Kd | 408 | — | |
HZZNLCVNOOMGDD
|
7.2 | IC50 | 2 | — | |
SPOWSXDVDODVEW
|
7.2 | IC50 | 2 | — | |
XSRHBCYNCKAFKS
|
7.2 | Ki | 45 | — | |
XUFLBSMTYMFOQH
|
7.2 | Ki | 43 | — | |
XZXHXSATPCNXJR
|
7.2 | Kd | 165 | Yes | |
ACXREQVXILYMKB
|
7.2 | IC50 | 3 | — | |
UJAUSTYSRUCHNY
|
7.2 | IC50 | 2 | — | |
WBSLEWFFUMKPFM
|
7.2 | IC50 | 2 | — | |
YOBIWCLAYQWPPW
|
7.2 | IC50 | 23 | — | |
JSFCBYKENXVGRL
|
7.2 | IC50 | 2 | — | |
OUJZYQBEFNDJQN
|
7.1 | Ki | 71 | — | |
XYXLUJQBBIBJFV
|
7.1 | Ki | 36 | — |