Target Details
| UniProt AC | P51812 |
|---|---|
| Gene Symbol | RPS6KA3 |
| Protein Name | Ribosomal protein S6 kinase alpha-3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 322
- Clinical molecules 28
- Avg pChEMBL 6.85
KEGG Pathways (10)
Associated Diseases (2)
Active Molecules (322)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YELZMARZEBVKBL
|
9.3 | Kd | 2 | — | |
KHGPYYFCIAISBU
|
9.0 | Ki | 31 | — | |
ZHMXXVNQAFCXKK
|
9.0 | IC50 | 15 | — | |
HKSZLNNOFSGOKW
|
8.8 | Ki | 118 | — | |
OSVUGUHRKMMBSE
|
8.7 | Kd | 170 | — | |
WKUUMSASAHOWGZ
|
8.7 | IC50 | 2 | — | |
VWVYILCFSYNJHF
|
8.6 | Ki | 49 | — | |
FCCMYBKAZCDQGX
|
8.5 | IC50 | 2 | — | |
XHCPCYVQXFHJAU
|
8.5 | IC50 | 12 | — | |
ZCCPLJOKGAACRT
|
8.4 | Kd | 599 | — | |
DTEKTGDVSARYDS
|
8.4 | IC50 | 3 | — | |
KJQYFARJBLRFQX
|
8.4 | IC50 | 3 | — | |
NXSJMRCTGYTSTK
|
8.4 | Kd | 200 | — | |
TWQIEMARYWIEFU
|
8.4 | IC50 | 2 | — | |
ADMFLILDQJSEIK
|
8.3 | Ki | 72 | — | |
IKUFKDGKRLMXEX
|
8.3 | IC50 | 3 | — | |
NWMPVMMGSHXANZ
|
8.3 | Ki | 58 | — | |
XYZNKCSDQRKAFR
|
8.3 | Ki | 53 | — | |
YUYJEQHNWKQNBT
|
8.3 | IC50 | 3 | — | |
DWRUMXZDNGCUDK
|
8.2 | IC50 | 3 | — | |
XYMNFMNOEWBPNB
|
8.2 | IC50 | 4 | — | |
NRGYMIVHSWOTKI
|
8.2 | IC50 | 2 | — | |
FYXRSVDHGLUMHB
|
8.2 | IC50 | 8 | — | |
MHGPJIHGGLSWFD
|
8.1 | IC50 | 8 | — | |
BQPLWJRDSDNGNE
|
8.1 | Ki | 16 | — | |
GHPFSYCYZJKVDZ
|
8.1 | Ki | 18 | Yes | |
VXYDJXMHISGSDA
|
8.1 | Ki | 59 | — | |
YWTBGJGMTBHQTM
|
8.1 | Ki | 65 | — | |
DSXXEELGXBCYNQ
|
8.0 | IC50 | 28 | Yes | |
ORUUEFDGYYTXAF
|
8.0 | Ki | 26 | — | |
OWRXHGAFWZFFCW
|
8.0 | Ki | 113 | — | |
RYYNGWLOYLRZLK
|
8.0 | Ki | 104 | — | |
XECUHDNZTMADFD
|
8.0 | IC50 | 2 | — | |
IEQAHFTVGLZUBI
|
8.0 | IC50 | 8 | — | |
LOLPPWBBNUVNQZ
|
8.0 | IC50 | 97 | Yes | |
IIRWNGPLJQXWFJ
|
7.9 | IC50 | 21 | — | |
KAKGFGCTONHQJW
|
7.9 | Ki | 25 | — | |
WDARYLSSWBWVCU
|
7.9 | Ki | 49 | — | |
YQKSNDNARJQAHP
|
7.9 | Ki | 12 | — | |
LAJAFFLJAJMYLK
|
7.9 | IC50 | 17 | — | |
IBUMAHMUIWPTCV
|
7.8 | IC50 | 3 | — | |
JGIBKTCCYJBOMS
|
7.8 | IC50 | 2 | — | |
IKLGYJACVCXYIL
|
7.8 | IC50 | 5 | — | |
PELFTNQHGSITLB
|
7.8 | IC50 | 2 | — | |
CHTMRWQLNNRRFJ
|
7.8 | Ki | 70 | — | |
NJPWCTYVEJIQBM
|
7.8 | Ki | 72 | — | |
UMTWTCVTRDYHQQ
|
7.8 | Ki | 56 | — | |
VIJBEUTVNBPGIU
|
7.8 | Ki | 19 | — | |
QQWUGDVOUVUTOY
|
7.8 | Kd | 231 | Yes | |
WMGGYIKBPUVPFM
|
7.8 | IC50 | 2 | — |