Target Details
| UniProt AC | P51787 |
|---|---|
| Gene Symbol | KCNQ1 |
| Protein Name | Potassium voltage-gated channel subfamily KQT member 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00520 (Ion_trans) PF03520 (KCNQ_channel) |
Summary
- Multi-target molecules 12
- Clinical molecules 0
- Avg pChEMBL 6.92
KEGG Pathways (6)
Associated Diseases (5)
Active Molecules (12)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XWQQRPSPOBDJLI
|
9.8 | IC50 | 40 | — | |
UFALWTGZIJAUPP
|
8.1 | IC50 | 3 | — | |
MSKWAZCFXKMVSS
|
7.3 | IC50 | 2 | — | |
SRZRLJWUQFIZRH
|
6.9 | IC50 | 2 | — | |
WHSNUPSZOQRQAB
|
6.7 | IC50 | 2 | — | |
SRZRLJWUQFIZRH
|
6.6 | IC50 | 2 | — | |
ICXASNQRNZTLLB
|
6.6 | IC50 | 2 | — | |
MSKWAZCFXKMVSS
|
6.4 | IC50 | 2 | — | |
SRZRLJWUQFIZRH
|
6.4 | IC50 | 2 | — | |
OHZDQMLJSUBQLE
|
6.2 | IC50 | 2 | — | |
QPWKXYZJANVPLF
|
6.1 | IC50 | 3 | — | |
WYJVNBJXXVCVIH
|
6.0 | IC50 | 2 | — |