Target Details
| UniProt AC | P51681 |
|---|---|
| Gene Symbol | CCR5 |
| Protein Name | C-C chemokine receptor type 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 126
- Clinical molecules 2
- Avg pChEMBL 7.38
KEGG Pathways (11)
- Chemokine signaling pathway
- Cytokine-cytokine receptor interaction
- Endocytosis
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- Kaposi sarcoma-associated herpesvirus infection
- Toxoplasmosis
- Viral carcinogenesis
- Viral life cycle - HIV-1
- Viral protein interaction with cytokine and cytokine receptor
- Virion - Human immunodeficiency virus
Associated Diseases (4)
Active Molecules (126)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NMYCPGLFRHGTSV
|
6.4 | IC50 | 2 | — | |
SSYDLAOTEQIPAM
|
6.4 | IC50 | 2 | — | |
XFUXIQVTGGYUOZ
|
6.4 | IC50 | 2 | — | |
MFORNGKVWCJAME
|
6.4 | IC50 | 2 | — | |
QYTDFOKICJWGHE
|
6.4 | IC50 | 2 | — | |
DSYMOXJOJWZVRV
|
6.4 | Ki | 2 | — | |
UUUTYZGDRKVSOB
|
6.4 | IC50 | 2 | — | |
COTMDVGGTIZRGD
|
6.3 | IC50 | 2 | — | |
DNPRHSLKGYTIJX
|
6.3 | IC50 | 2 | — | |
LRWWYYRQZRJLHU
|
6.3 | IC50 | 2 | — | |
DSWXTSLXHOCGMH
|
6.2 | IC50 | 2 | — | |
YLVBQGLIQXQGPH
|
6.2 | IC50 | 2 | — | |
OIGUMNDUYFBXEM
|
6.2 | IC50 | 3 | — | |
UAKDPJAUOVRMIX
|
6.2 | IC50 | 2 | — | |
XTBMGQICBMRHTA
|
6.2 | IC50 | 2 | — | |
AWEGVPOPWDMWCC
|
6.2 | IC50 | 2 | — | |
VQNLJXWZGVRLBA
|
6.2 | IC50 | 2 | — | |
IUENSEDRGKTRGA
|
6.1 | IC50 | 2 | — | |
GVOISEJVFFIGQE
|
6.1 | IC50 | 2 | — | |
WLNCGIQLHPVTPW
|
6.1 | IC50 | 3 | Yes | |
FLINZDKAJGFTLP
|
6.1 | IC50 | 2 | — | |
GUGOEEXESWIERI
|
6.1 | Ki | 18 | Yes | |
BXCVNDLGUWFNBK
|
6.0 | IC50 | 2 | — | |
DNPRHSLKGYTIJX
|
6.0 | IC50 | 2 | — | |
HEXTXRMVMKIBQR
|
6.0 | IC50 | 3 | — | |
NDZYPHLNJZSQJY
|
6.0 | IC50 | 3 | — |