Target Details
| UniProt AC | P51681 |
|---|---|
| Gene Symbol | CCR5 |
| Protein Name | C-C chemokine receptor type 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 126
- Clinical molecules 2
- Avg pChEMBL 7.38
KEGG Pathways (11)
- Chemokine signaling pathway
- Cytokine-cytokine receptor interaction
- Endocytosis
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- Kaposi sarcoma-associated herpesvirus infection
- Toxoplasmosis
- Viral carcinogenesis
- Viral life cycle - HIV-1
- Viral protein interaction with cytokine and cytokine receptor
- Virion - Human immunodeficiency virus
Associated Diseases (4)
Active Molecules (126)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MMFPYPNUFANCKT
|
7.6 | IC50 | 2 | — | |
UUUTYZGDRKVSOB
|
7.5 | Ki | 2 | — | |
OPHYHBRVLAQKEG
|
7.5 | IC50 | 3 | — | |
QLVOILJNRVKKRP
|
7.5 | IC50 | 2 | — | |
DECZUBPHXAXNSH
|
7.5 | Ki | 2 | — | |
RAKTXXNBDRXTAX
|
7.5 | Ki | 2 | — | |
SWXHHKZYRFCOPH
|
7.5 | Ki | 2 | — | |
QRKQGOWSACQLGK
|
7.5 | IC50 | 2 | — | |
RFNTZDWBOZXHTR
|
7.5 | IC50 | 2 | — | |
QAPTWHXHEYAIKG
|
7.5 | IC50 | 2 | — | |
YJGRIVQJUHTIGN
|
7.5 | IC50 | 2 | — | |
ZHSPLCRKVQNOGM
|
7.4 | IC50 | 2 | — | |
XYCUIMUECGHTFV
|
7.3 | Ki | 2 | — | |
CSTRIVMEIYPLGJ
|
7.3 | Ki | 2 | — | |
DTYWPXSMHVEQQW
|
7.2 | IC50 | 2 | — | |
FCBWQXORDQYHFI
|
7.2 | IC50 | 2 | — | |
YLNOGPJREAMGJN
|
7.2 | IC50 | 2 | — | |
YEQJVHQCUDMXFG
|
7.2 | Ki | 2 | — | |
TWDSSLGDUOHXCF
|
7.1 | IC50 | 3 | — | |
NMYCPGLFRHGTSV
|
7.1 | IC50 | 2 | — | |
KLBHHUODQVCBKX
|
7.1 | IC50 | 2 | — | |
CWRFGTWBBWBDRR
|
7.0 | IC50 | 2 | — | |
DFPLYLKKYSEABD
|
7.0 | IC50 | 2 | — | |
YWUQJCUUNVCNFS
|
7.0 | IC50 | 2 | — | |
NMYCPGLFRHGTSV
|
7.0 | IC50 | 2 | — | |
WKTVEPAXEKXDKZ
|
7.0 | IC50 | 2 | — | |
FVNQVTADUDKSGZ
|
6.9 | IC50 | 2 | — | |
BAVVASQPMQMZER
|
6.9 | IC50 | 2 | — | |
BAVVASQPMQMZER
|
6.9 | IC50 | 2 | — | |
IDSHXLDGGWIGBW
|
6.9 | IC50 | 2 | — | |
OKIJQELRSBSEJX
|
6.9 | IC50 | 2 | — | |
SNVMTABEFLKIEG
|
6.8 | IC50 | 2 | — | |
HKIFMAJLMSGIOP
|
6.8 | Ki | 2 | — | |
CJGHKRWUTQLMOP
|
6.7 | IC50 | 2 | — | |
DSWXTSLXHOCGMH
|
6.7 | IC50 | 2 | — | |
PEFVTWREQBVUOK
|
6.7 | IC50 | 2 | — | |
VBMPRCMEFUCQPO
|
6.7 | IC50 | 2 | — | |
FFBYNQCXDQNNQT
|
6.7 | Ki | 2 | — | |
BXZCHELXYNXCDS
|
6.7 | IC50 | 2 | — | |
LFEZDWBBQLHEMC
|
6.7 | IC50 | 2 | — | |
VSAYPYFFICXMGV
|
6.6 | Ki | 2 | — | |
GQLXQNMFKWOOSD
|
6.6 | IC50 | 3 | — | |
CHNSDJOKVUZBQF
|
6.6 | IC50 | 2 | — | |
AOPWQMZXHFQASV
|
6.5 | IC50 | 2 | — | |
PJTGSIKANITYOO
|
6.5 | IC50 | 2 | — | |
DNPRHSLKGYTIJX
|
6.5 | IC50 | 2 | — | |
NTTROUGKGFNVGR
|
6.5 | IC50 | 2 | — | |
BYVKUTDQYZLLAZ
|
6.5 | IC50 | 2 | — | |
SCSTUPQPTWXCHZ
|
6.5 | IC50 | 2 | — | |
HTWLSEXOVXEWKJ
|
6.5 | Ki | 2 | — |