Target Details
| UniProt AC | P51679 |
|---|---|
| Gene Symbol | CCR4 |
| Protein Name | C-C chemokine receptor type 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 22
- Clinical molecules 0
- Avg pChEMBL 6.71
KEGG Pathways (5)
Active Molecules (22)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HDQNDRCZSVEGSG
|
8.1 | IC50 | 5 | — | |
JBBKREGWJICILL
|
8.1 | IC50 | 5 | — | |
SPLGZZDGUQTEHE
|
8.0 | IC50 | 5 | — | |
DGPHJNJINCRCKW
|
7.4 | IC50 | 5 | — | |
YTEVTHHGQMUPHC
|
7.4 | IC50 | 2 | — | |
KBLOFZHBIDLNIS
|
7.0 | IC50 | 5 | — | |
KCVWGCOBGFLUEB
|
6.9 | IC50 | 5 | — | |
RIEUAZKSQUTJQU
|
6.8 | Ki | 3 | — | |
UFZMURFKAOEOKB
|
6.5 | IC50 | 2 | — | |
HZPZDNAFDLIEJH
|
6.4 | Ki | 3 | — | |
OIGUMNDUYFBXEM
|
6.4 | Ki | 3 | — | |
YGWURLOZYUXZKA
|
6.4 | Ki | 5 | — | |
ZHOSAEFOHKXJDJ
|
6.3 | IC50 | 5 | — | |
HILQSLVIBNFOMC
|
6.3 | IC50 | 2 | — | |
DRHNPWMFAGWFPG
|
6.3 | Ki | 3 | — | |
VZPTWPGJCWIVGK
|
6.3 | Ki | 2 | — | |
NAYZSSQGIKJDGG
|
6.2 | IC50 | 2 | — | |
DLTXTHJGLDWETN
|
6.2 | Ki | 2 | — | |
YSVHPACWAGFQQP
|
6.2 | Ki | 3 | — | |
GQLXQNMFKWOOSD
|
6.1 | Ki | 3 | — | |
CDGRGHROXAGDDT
|
6.0 | Ki | 2 | — | |
GMFHGEGAYGJWAD
|
6.0 | Ki | 2 | — |