Target Details
| UniProt AC | P51677 |
|---|---|
| Gene Symbol | CCR3 |
| Protein Name | C-C chemokine receptor type 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 221
- Clinical molecules 0
- Avg pChEMBL 8.05
KEGG Pathways (6)
Active Molecules (221)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RECBRJKCPMUFRD
|
9.9 | IC50 | 2 | — | |
AYPGYVOWMUSFPT
|
9.7 | Ki | 2 | — | |
IQUQYZRIYXKKDB
|
9.7 | IC50 | 2 | — | |
NZFSPDVTABQASR
|
9.5 | Ki | 3 | — | |
YXGHCLLTAXLPMG
|
9.4 | IC50 | 2 | — | |
RKHFLVYZXJYWKW
|
9.3 | IC50 | 4 | — | |
SEIOTCVWLCUESB
|
9.3 | Ki | 2 | — | |
WKNWCTUFTMDACE
|
9.3 | Ki | 2 | — | |
VQHKDCUXFKNNMT
|
9.2 | IC50 | 2 | — | |
HEXTXRMVMKIBQR
|
9.2 | IC50 | 3 | — | |
YVVCYGCCIFEDCL
|
9.2 | IC50 | 2 | — | |
HFWLILWGBZWYRI
|
9.2 | Ki | 2 | — | |
NDZYPHLNJZSQJY
|
9.2 | IC50 | 3 | — | |
NNOWQHZNUGOGEV
|
9.2 | IC50 | 3 | — | |
TXFKRSLQBDPWHK
|
9.2 | IC50 | 2 | — | |
GWVFJNPANMKQSY
|
9.1 | Ki | 2 | — | |
IBTMKWBYOYIWBF
|
9.1 | Ki | 2 | — | |
JPDUMUHTXIBGHJ
|
9.1 | Ki | 3 | — | |
KDBCNKHHBUKNRH
|
9.1 | IC50 | 2 | — | |
YDHQRFQQOKRWAD
|
9.1 | Ki | 2 | — | |
FRPOMOOESVDDAO
|
9.1 | IC50 | 2 | — | |
FTVCCHUPUJEUIW
|
9.1 | IC50 | 4 | — | |
KHIUUVSTTUGPRZ
|
9.1 | IC50 | 3 | — | |
HTZBCHVAMWNYJY
|
9.0 | IC50 | 2 | — | |
JMTZNRURKTUFTP
|
9.0 | IC50 | 2 | — | |
UHVITKONHRHSFJ
|
9.0 | IC50 | 4 | — | |
YMYZSITWBGWUAF
|
9.0 | Ki | 2 | — | |
RRHZFCXDULLQHS
|
8.9 | IC50 | 2 | — | |
KLUPWQNJJYFUHQ
|
8.9 | IC50 | 2 | — | |
LVNMVTRHDJLKCU
|
8.9 | IC50 | 2 | — | |
SPDRJYHRLHGQBR
|
8.9 | IC50 | 2 | — | |
XLKVTYHUNRLGJS
|
8.9 | IC50 | 2 | — | |
ASRDPULQBHFPGU
|
8.9 | IC50 | 7 | — | |
DLONTNINHYMHFB
|
8.9 | Ki | 2 | — | |
GEMBQNHUTJFAFL
|
8.9 | Ki | 2 | — | |
LEHDCEDFGAFVGX
|
8.9 | Ki | 2 | — | |
ZSHFBVRJUAGORQ
|
8.9 | IC50 | 4 | — | |
GHILKFUWMODLTJ
|
8.8 | IC50 | 2 | — | |
WYKUNXLKNJTHND
|
8.8 | IC50 | 4 | — | |
WKMAJEHBPREIER
|
8.8 | IC50 | 2 | — | |
NBEYIKPRTIBJBG
|
8.8 | IC50 | 2 | — | |
NDXPOARUSJMOJN
|
8.8 | Ki | 2 | — | |
RGQXJYRGDMABLT
|
8.8 | Ki | 3 | — | |
TYDWSEQLTIBAPO
|
8.8 | Ki | 2 | — | |
XBJQRDCFABQBGT
|
8.8 | Ki | 3 | — | |
YSQQOGOBORIIMG
|
8.8 | Ki | 2 | — | |
CTZCYZCFMJXNPE
|
8.8 | IC50 | 2 | — | |
JJILEQNLSXCPPS
|
8.8 | IC50 | 2 | — | |
SLSRYMJCMOWUIE
|
8.8 | IC50 | 4 | — | |
OIXSYJAHIPQFMO
|
8.7 | Ki | 2 | — |