Target Details
| UniProt AC | P51617 |
|---|---|
| Gene Symbol | IRAK1 |
| Protein Name | Interleukin-1 receptor-associated kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00531 (Death) PF00069 (Pkinase) |
Summary
- Multi-target molecules 312
- Clinical molecules 15
- Avg pChEMBL 6.84
KEGG Pathways (20)
- Alcoholic liver disease
- Chagas disease
- Coronavirus disease - COVID-19
- Epstein-Barr virus infection
- Hepatitis B
- Herpes simplex virus 1 infection
- Human immunodeficiency virus 1 infection
- Leishmaniasis
- Lipid and atherosclerosis
- MAPK signaling pathway
- Measles
- NF-kappa B signaling pathway
- Neurotrophin signaling pathway
- Pathogenic Escherichia coli infection
- Pertussis
- Salmonella infection
- Toll-like receptor signaling pathway
- Toxoplasmosis
- Tuberculosis
- Yersinia infection
Active Molecules (312)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QAJPIJHWTGPUNZ
|
6.8 | Ki | 37 | — | |
WRDPDAIOMMMLNR
|
6.8 | IC50 | 2 | — | |
MURKOANUFGPGGP
|
6.8 | IC50 | 2 | — | |
PIQCTGMSNWUMAF
|
6.8 | Kd | 137 | Yes | |
WPXVVAWAHQHJPF
|
6.8 | IC50 | 41 | — | |
FEJCKYYKSNIWCL
|
6.7 | Ki | 2 | — | |
WGQUSQTWZRXHGK
|
6.7 | IC50 | 3 | — | |
ZRZMENVDJBJBOY
|
6.7 | IC50 | 3 | — | |
APNCLDVFDSDLCS
|
6.7 | IC50 | 2 | — | |
KTEIFNKAUNYNJU
|
6.7 | Ki | 48 | — | |
UJFKYOVASOKVMM
|
6.7 | IC50 | 2 | — | |
GJMNFLBPIHSIRV
|
6.7 | IC50 | 2 | — | |
MXCUSZDSXDTMHC
|
6.7 | IC50 | 3 | — | |
CRSHGUZUNKJVIT
|
6.7 | IC50 | 2 | — | |
GUBJNPWVIUFSTR
|
6.7 | Kd | 103 | — | |
JOOXLOJCABQBSG
|
6.7 | Kd | 139 | — | |
TZUYQGIZCUHALE
|
6.7 | IC50 | 2 | — | |
MJGKLMMMXSNBCX
|
6.7 | IC50 | 3 | — | |
ULXXDDBFHOBEHA
|
6.6 | Kd | 15 | Yes | |
CMJCXYNUCSMDBY
|
6.6 | Kd | 15 | — | |
XPMRQKGHVCXNDM
|
6.6 | IC50 | 2 | — | |
AOFJRBMLTUGMMP
|
6.6 | Ki | 12 | — | |
LYNBNVBMAGDJRW
|
6.6 | Ki | 81 | — | |
SBFPHSVZEXSHTL
|
6.6 | Ki | 62 | — | |
YWTBGJGMTBHQTM
|
6.6 | Ki | 65 | — | |
DYNHJHQFHQTFTP
|
6.6 | Kd | 38 | — | |
PDXCPPIXNVTKCI
|
6.6 | IC50 | 2 | — | |
HFNKQEVNSGCOJV
|
6.5 | Kd | 65 | — | |
BPTXXXCWMKGAFJ
|
6.5 | IC50 | 2 | — | |
NXSJMRCTGYTSTK
|
6.5 | Kd | 200 | — | |
QTCFYQHZJIIHBS
|
6.5 | IC50 | 2 | — | |
WHCMKDGCCYRJKV
|
6.5 | IC50 | 2 | — | |
ZXPBSKBKOLENLI
|
6.5 | IC50 | 2 | — | |
HEUSUIRCBWROMH
|
6.5 | Ki | 64 | — | |
JJJSCYSPSKBQAX
|
6.5 | Ki | 34 | — | |
NRSGWEVTVGZDFC
|
6.5 | Ki | 50 | — | |
OADRBDVURCEKRP
|
6.5 | Ki | 44 | — | |
UMTWTCVTRDYHQQ
|
6.5 | Ki | 56 | — | |
ZVWRFVCNQOECJS
|
6.5 | Ki | 71 | — | |
PFCFMZHQWUDEEB
|
6.5 | Ki | 2 | — | |
LBBNQAJEJZYWPT
|
6.4 | IC50 | 2 | — | |
DIZQXPLWZKQART
|
6.4 | IC50 | 2 | — | |
IEOZVBDPTHRYGK
|
6.4 | Ki | 3 | — | |
HHCBMISMPSAZBF
|
6.4 | IC50 | 23 | — | |
CEAYRKIZESVQSN
|
6.4 | Ki | 4 | — | |
IOBVCHJTLVPPBR
|
6.4 | Ki | 39 | — | |
PSBLEKZDHVNIQM
|
6.4 | Ki | 2 | — | |
RTDSHUGNRVXRHN
|
6.4 | Ki | 51 | — | |
XOVPCPRZRHQFBI
|
6.4 | Ki | 15 | — | |
DKZYXHCYPUVGAF
|
6.4 | Kd | 112 | — |